Discovery of 1-Amino-1H-imidazole-5-carboxamide Derivatives as Highly Selective, Covalent Bruton's Tyrosine Kinase (BTK) Inhibitors.
Ma C, Li Q, Zhao M, Fan G, Zhao J, Zhang D, Yang S, Zhang S, Gao D, Mao L, Zhu L, Li W, Xu G, Jiang Y, Ding Q.
Ma C, et al. Among authors: zhang s, zhang d.
J Med Chem. 2021 Nov 11;64(21):16242-16270. doi: 10.1021/acs.jmedchem.1c01559. Epub 2021 Oct 21.
J Med Chem. 2021.
PMID: 34672559