Proschak E - Search Results

1

Phosphatase activity of soluble epoxide hydrolase.

Kramer J, Proschak E. Kramer J, et al. Among authors: proschak e. Prostaglandins Other Lipid Mediat. 2017 Nov;133:88-92. doi: 10.1016/j.prostaglandins.2017.07.002. Epub 2017 Jul 17. Prostaglandins Other Lipid Mediat. 2017. PMID: 28729091 Review.

2

Complementary screening techniques yielded fragments that inhibit the phosphatase activity of soluble epoxide hydrolase.

Hahn S, Achenbach J, Buscató E, Klingler FM, Schroeder M, Meirer K, Hieke M, Heering J, Barbosa-Sicard E, Loehr F, Fleming I, Doetsch V, Schubert-Zsilavecz M, Steinhilber D, Proschak E. Hahn S, et al. Among authors: proschak e. ChemMedChem. 2011 Dec 9;6(12):2146-9. doi: 10.1002/cmdc.201100433. Epub 2011 Oct 21. ChemMedChem. 2011. PMID: 22021219 No abstract available.

3

Evaluation of structure-derived pharmacophore of soluble epoxide hydrolase inhibitors by virtual screening.

Moser D, Achenbach J, Klingler FM, Estel la B, Hahn S, Proschak E. Moser D, et al. Among authors: proschak e. Bioorg Med Chem Lett. 2012 Nov 1;22(21):6762-5. doi: 10.1016/j.bmcl.2012.08.066. Epub 2012 Aug 23. Bioorg Med Chem Lett. 2012. PMID: 23017883

4

Design and synthesis of dual modulators of soluble epoxide hydrolase and peroxisome proliferator-activated receptors.

la Buscató E, Blöcher R, Lamers C, Klingler FM, Hahn S, Steinhilber D, Schubert-Zsilavecz M, Proschak E. la Buscató E, et al. Among authors: proschak e. J Med Chem. 2012 Dec 13;55(23):10771-5. doi: 10.1021/jm301194c. Epub 2012 Nov 19. J Med Chem. 2012. PMID: 23130964

5

Synthesis and structure-activity relationship studies of novel dual inhibitors of soluble epoxide hydrolase and 5-lipoxygenase.

Meirer K, Rödl CB, Wisniewska JM, George S, Häfner AK, Buscató EL, Klingler FM, Hahn S, Berressem D, Wittmann SK, Steinhilber D, Hofmann B, Proschak E. Meirer K, et al. Among authors: proschak e. J Med Chem. 2013 Feb 28;56(4):1777-81. doi: 10.1021/jm301617j. Epub 2013 Feb 7. J Med Chem. 2013. PMID: 23356879

6

From a multipotent stilbene to soluble epoxide hydrolase inhibitors with antiproliferative properties.

Buscató E, Büttner D, Brüggerhoff A, Klingler FM, Weber J, Scholz B, Zivković A, Marschalek R, Stark H, Steinhilber D, Bode HB, Proschak E. Buscató E, et al. Among authors: proschak e. ChemMedChem. 2013 Jun;8(6):919-23. doi: 10.1002/cmdc.201300057. Epub 2013 Apr 17. ChemMedChem. 2013. PMID: 23596124

7

PENG: a neural gas-based approach for pharmacophore elucidation. method design, validation, and virtual screening for novel ligands of LTA4H.

Moser D, Wittmann SK, Kramer J, Blöcher R, Achenbach J, Pogoryelov D, Proschak E. Moser D, et al. Among authors: proschak e. J Chem Inf Model. 2015 Feb 23;55(2):284-93. doi: 10.1021/ci500618u. Epub 2015 Feb 9. J Chem Inf Model. 2015. PMID: 25625859

8

N-Benzylbenzamides: A Novel Merged Scaffold for Orally Available Dual Soluble Epoxide Hydrolase/Peroxisome Proliferator-Activated Receptor γ Modulators.

Blöcher R, Lamers C, Wittmann SK, Merk D, Hartmann M, Weizel L, Diehl O, Brüggerhoff A, Boß M, Kaiser A, Schader T, Göbel T, Grundmann M, Angioni C, Heering J, Geisslinger G, Wurglics M, Kostenis E, Brüne B, Steinhilber D, Schubert-Zsilavecz M, Kahnt AS, Proschak E. Blöcher R, et al. Among authors: proschak e. J Med Chem. 2016 Jan 14;59(1):61-81. doi: 10.1021/acs.jmedchem.5b01239. Epub 2015 Dec 25. J Med Chem. 2016. PMID: 26595749

9

Bacterial Expression and HTS Assessment of Soluble Epoxide Hydrolase Phosphatase.

Klingler FM, Wolf M, Wittmann S, Gribbon P, Proschak E. Klingler FM, et al. Among authors: proschak e. J Biomol Screen. 2016 Aug;21(7):689-94. doi: 10.1177/1087057116637609. Epub 2016 Mar 23. J Biomol Screen. 2016. PMID: 27009944

10

Thermodynamic properties of leukotriene A₄ hydrolase inhibitors.

Wittmann SK, Kalinowsky L, Kramer JS, Bloecher R, Knapp S, Steinhilber D, Pogoryelov D, Proschak E, Heering J. Wittmann SK, et al. Among authors: proschak e. Bioorg Med Chem. 2016 Nov 1;24(21):5243-5248. doi: 10.1016/j.bmc.2016.08.047. Epub 2016 Aug 26. Bioorg Med Chem. 2016. PMID: 27651294

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