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pH-dependent ileocolonic drug delivery, part II: preclinical evaluation of novel drugs and novel excipients.
Drug Discov Today. 2020 Aug;25(8):1374-1388. doi: 10.1016/j.drudis.2020.06.012. Epub 2020 Jun 17.
Drug Discov Today. 2020.
PMID: 32562842
Free article.
Review.
pH-dependent ileocolonic drug delivery, part I: in vitro and clinical evaluation of novel systems.
Broesder A, Woerdenbag HJ, Prins GH, Nguyen DN, Frijlink HW, Hinrichs WLJ.
Broesder A, et al.
Drug Discov Today. 2020 Aug;25(8):1362-1373. doi: 10.1016/j.drudis.2020.06.011. Epub 2020 Jun 15.
Drug Discov Today. 2020.
PMID: 32554060
Free article.
Review.
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Ileo-Colon Targeting of the Poorly Water-Soluble Drug Celecoxib Using a pH-Dependent Coating in Combination with Self-Emulsifying Drug Delivery or Solid Dispersion Systems.
Broesder A, Berends JME, Scheepers SM, Nguyen DN, Frijlink HW, Hinrichs WLJ.
Broesder A, et al.
Pharmaceutics. 2021 May 15;13(5):731. doi: 10.3390/pharmaceutics13050731.
Pharmaceutics. 2021.
PMID: 34063521
Free PMC article.
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Formulation and In Vitro Evaluation of Pellets Containing Sulfasalazine and Caffeine to Verify Ileo-Colonic Drug Delivery.
Broesder A, Bircan SY, de Waard AB, Eissens AC, Frijlink HW, Hinrichs WLJ.
Broesder A, et al.
Pharmaceutics. 2021 Nov 23;13(12):1985. doi: 10.3390/pharmaceutics13121985.
Pharmaceutics. 2021.
PMID: 34959267
Free PMC article.
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Polymeric microspheres for the sustained release of a protein-based drug carrier targeting the PDGFβ-receptor in the fibrotic kidney.
Teekamp N, Van Dijk F, Broesder A, Evers M, Zuidema J, Steendam R, Post E, Hillebrands JL, Frijlink HW, Poelstra K, Beljaars L, Olinga P, Hinrichs WLJ.
Teekamp N, et al. Among authors: broesder a.
Int J Pharm. 2017 Dec 20;534(1-2):229-236. doi: 10.1016/j.ijpharm.2017.09.072. Epub 2017 Oct 14.
Int J Pharm. 2017.
PMID: 29038068
Free article.
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