Zessin M - Search Results

1

Key structural requirements of benzamide derivatives for histone deacetylase inhibition: design, synthesis and biological evaluation.

Cheshmazar N, Hamzeh-Mivehroud M, Hemmati S, Abolhasani H, Heidari F, Charoudeh HN, Zessin M, Schutkowski M, Sippl W, Dastmalchi S. Cheshmazar N, et al. Among authors: zessin m. Future Med Chem. 2024 Apr 16. doi: 10.4155/fmc-2023-0122. Online ahead of print. Future Med Chem. 2024. PMID: 38623995

2

Application of Ligand- and Structure-Based Prediction Models for the Design of Alkylhydrazide-Based HDAC3 Inhibitors as Novel Anti-Cancer Compounds.

Bülbül EF, Robaa D, Sun P, Mahmoudi F, Melesina J, Zessin M, Schutkowski M, Sippl W. Bülbül EF, et al. Among authors: zessin m. Pharmaceuticals (Basel). 2023 Jul 6;16(7):968. doi: 10.3390/ph16070968. Pharmaceuticals (Basel). 2023. PMID: 37513880 Free PMC article.

3

Novel hydroxamic acid derivative induces apoptosis and constrains autophagy in leukemic cells.

Fischer MA, Mustafa AM, Hausmann K, Ashry R, Kansy AG, Liebl MC, Brachetti C, Piée-Staffa A, Zessin M, Ibrahim HS, Hofmann TG, Schutkowski M, Sippl W, Krämer OH. Fischer MA, et al. Among authors: zessin m. J Adv Res. 2023 Jul 17:S2090-1232(23)00197-2. doi: 10.1016/j.jare.2023.07.005. Online ahead of print. J Adv Res. 2023. PMID: 37467961 Free article.

4

Continuous Fluorescent Sirtuin Activity Assay Based on Fatty Acylated Lysines.

Zessin M, Meleshin M, Hilscher S, Schiene-Fischer C, Barinka C, Jung M, Schutkowski M. Zessin M, et al. Int J Mol Sci. 2023 Apr 18;24(8):7416. doi: 10.3390/ijms24087416. Int J Mol Sci. 2023. PMID: 37108579 Free PMC article.

5

Development of Alkylated Hydrazides as Highly Potent and Selective Class I Histone Deacetylase Inhibitors with T cell Modulatory Properties.

Sun P, Wang J, Khan KS, Yang W, Ng BW, Ilment N, Zessin M, Bülbül EF, Robaa D, Erdmann F, Schmidt M, Romier C, Schutkowski M, Cheng AS, Sippl W. Sun P, et al. Among authors: zessin m. J Med Chem. 2022 Dec 22;65(24):16313-16337. doi: 10.1021/acs.jmedchem.2c01132. Epub 2022 Nov 30. J Med Chem. 2022. PMID: 36449385

6

Continuous Histone Deacylase Activity Assays.

Zessin M, Meleshin M, Sippl W, Schutkowski M. Zessin M, et al. Methods Mol Biol. 2023;2589:411-428. doi: 10.1007/978-1-0716-2788-4_27. Methods Mol Biol. 2023. PMID: 36255640

7

Development of Pyrazine-Anilinobenzamides as Histone Deacetylase HDAC1-3 Selective Inhibitors and Biological Testing Against Pancreas Cancer Cell Lines.

Abdelsalam M, Ibrahim HS, Krauss L, Zessin M, Vecchio A, Hastreiter S, Schutkowski M, Schneider G, Sippl W. Abdelsalam M, et al. Among authors: zessin m. Methods Mol Biol. 2023;2589:145-155. doi: 10.1007/978-1-0716-2788-4_10. Methods Mol Biol. 2023. PMID: 36255623

8

Small Changes Make the Difference for SIRT2: Two Different Binding Modes for 3-Arylmercapto-Acylated Lysine Derivatives.

Kalbas D, Meleshin M, Liebscher S, Zessin M, Melesina J, Schiene-Fischer C, Bülbül EF, Bordusa F, Sippl W, Schutkowski M. Kalbas D, et al. Among authors: zessin m. Biochemistry. 2022 Sep 6;61(17):1705-1722. doi: 10.1021/acs.biochem.2c00211. Epub 2022 Aug 16. Biochemistry. 2022. PMID: 35972884

9

Uncovering Robust Delactoylase and Depyruvoylase Activities of HDAC Isoforms.

Zessin M, Meleshin M, Praetorius L, Sippl W, Bařinka C, Schutkowski M. Zessin M, et al. ACS Chem Biol. 2022 Jun 17;17(6):1364-1375. doi: 10.1021/acschembio.1c00863. Epub 2022 May 31. ACS Chem Biol. 2022. PMID: 35639992

10

Development of New Inhibitors of HDAC1-3 Enzymes Aided by In Silico Design Strategies.

Cheshmazar N, Hemmati S, Hamzeh-Mivehroud M, Sokouti B, Zessin M, Schutkowski M, Sippl W, Nozad Charoudeh H, Dastmalchi S. Cheshmazar N, et al. Among authors: zessin m. J Chem Inf Model. 2022 May 23;62(10):2387-2397. doi: 10.1021/acs.jcim.1c01557. Epub 2022 Apr 25. J Chem Inf Model. 2022. PMID: 35467871

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