Sugasawa K - Search Results

1

Improved Dose-Response Relationship of (+)-Discodermolide-Taxol Hybrid Congeners.

Nadaradjane C, Yang CH, Rodriguez-Gabin A, Ye K, Sugasawa K, Atasoylu O, Smith AB 3rd, Horwitz SB, McDaid HM. Nadaradjane C, et al. Among authors: sugasawa k. J Nat Prod. 2018 Mar 23;81(3):607-615. doi: 10.1021/acs.jnatprod.8b00111. Epub 2018 Mar 9. J Nat Prod. 2018. PMID: 29522336 Free PMC article.

2

Design and synthesis of (+)-discodermolide-paclitaxel hybrids leading to enhanced biological activity.

Smith AB, Sugasawa K, Atasoylu O, Yang CP, Horwitz SB. Smith AB, et al. Among authors: sugasawa k. J Med Chem. 2011 Sep 22;54(18):6319-27. doi: 10.1021/jm200692n. Epub 2011 Aug 26. J Med Chem. 2011. PMID: 21870795 Free PMC article.

3

Direct modulation of microtubule stability contributes to anthracene general anesthesia.

Emerson DJ, Weiser BP, Psonis J, Liao Z, Taratula O, Fiamengo A, Wang X, Sugasawa K, Smith AB 3rd, Eckenhoff RG, Dmochowski IJ. Emerson DJ, et al. Among authors: sugasawa k. J Am Chem Soc. 2013 Apr 10;135(14):5389-98. doi: 10.1021/ja311171u. Epub 2013 Mar 29. J Am Chem Soc. 2013. PMID: 23484901 Free PMC article.

4

Discovery of N-[2-hydroxy-6-(4-methoxybenzamido)phenyl]-4- (4-methyl-1,4-diazepan-1-yl)benzamide (darexaban, YM150) as a potent and orally available factor Xa inhibitor.

Hirayama F, Koshio H, Ishihara T, Hachiya S, Sugasawa K, Koga Y, Seki N, Shiraki R, Shigenaga T, Iwatsuki Y, Moritani Y, Mori K, Kadokura T, Kawasaki T, Matsumoto Y, Sakamoto S, Tsukamoto S. Hirayama F, et al. Among authors: sugasawa k. J Med Chem. 2011 Dec 8;54(23):8051-65. doi: 10.1021/jm200868m. Epub 2011 Nov 11. J Med Chem. 2011. PMID: 21995444

5

Synthesis and structure-activity relationships of a series of benzazepine derivatives as 5-HT2C receptor agonists.

Shimada I, Maeno K, Kondoh Y, Kaku H, Sugasawa K, Kimura Y, Hatanaka K, Naitou Y, Wanibuchi F, Sakamoto S, Tsukamoto S. Shimada I, et al. Among authors: sugasawa k. Bioorg Med Chem. 2008 Mar 15;16(6):3309-20. doi: 10.1016/j.bmc.2007.12.009. Epub 2007 Dec 8. Bioorg Med Chem. 2008. PMID: 18083579

6

Pharmacological profile of AS1670542, a novel orally-active human thrombopoietin receptor agonist.

Abe M, Suzuki K, Sakata C, Sugasawa K, Hirayama F, Koga Y, Kawasaki T, Naganuma S, Itoh H. Abe M, et al. Among authors: sugasawa k. Eur J Pharmacol. 2011 Jan 10;650(1):58-63. doi: 10.1016/j.ejphar.2010.09.072. Epub 2010 Oct 13. Eur J Pharmacol. 2011. PMID: 20950606

7

Novel strategy to boost oral anticoagulant activity of blood coagulation enzyme inhibitors based on biotransformation into hydrophilic conjugates.

Ishihara T, Koga Y, Mori K, Sugasawa K, Iwatsuki Y, Hirayama F. Ishihara T, et al. Among authors: sugasawa k. Bioorg Med Chem. 2014 Nov 15;22(22):6324-32. doi: 10.1016/j.bmc.2014.09.059. Epub 2014 Oct 19. Bioorg Med Chem. 2014. PMID: 25438755

8

AKR-501 (YM477) a novel orally-active thrombopoietin receptor agonist.

Fukushima-Shintani M, Suzuki K, Iwatsuki Y, Abe M, Sugasawa K, Hirayama F, Kawasaki T, Nakahata T. Fukushima-Shintani M, et al. Among authors: sugasawa k. Eur J Haematol. 2009 Apr;82(4):247-54. doi: 10.1111/j.1600-0609.2008.01198.x. Epub 2009 Jan 16. Eur J Haematol. 2009. PMID: 19183407

9

AKR-501 (YM477) in combination with thrombopoietin enhances human megakaryocytopoiesis.

Fukushima-Shintani M, Suzuki K, Iwatsuki Y, Abe M, Sugasawa K, Hirayama F, Kawasaki T. Fukushima-Shintani M, et al. Among authors: sugasawa k. Exp Hematol. 2008 Oct;36(10):1337-42. doi: 10.1016/j.exphem.2008.04.020. Epub 2008 Jul 10. Exp Hematol. 2008. PMID: 18619724 Free article.

10

The effect of self-management vestibular rehabilitation on persistent postural-perceptual dizziness.

Fujimoto C, Oka M, Ichijo K, Kinoshita M, Kamogashira T, Sugasawa K, Kawahara T, Yamasoba T. Fujimoto C, et al. Among authors: sugasawa k. Laryngoscope Investig Otolaryngol. 2023 May 29;8(4):1014-1020. doi: 10.1002/lio2.1073. eCollection 2023 Aug. Laryngoscope Investig Otolaryngol. 2023. PMID: 37621292 Free PMC article.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

194 results

Search Page