Staszewski M - Search Results

1

Search for multifunctional agents against Alzheimer's disease among non-imidazole histamine H3 receptor ligands. In vitro and in vivo pharmacological evaluation and computational studies of piperazine derivatives.

Jończyk J, Lodarski K, Staszewski M, Godyń J, Zaręba P, Soukup O, Janockova J, Korabecny J, Sałat K, Malikowska-Racia N, Hebda M, Szałaj N, Filipek B, Walczyński K, Malawska B, Bajda M. Jończyk J, et al. Among authors: staszewski m. Bioorg Chem. 2019 Sep;90:103084. doi: 10.1016/j.bioorg.2019.103084. Epub 2019 Jun 26. Bioorg Chem. 2019. PMID: 31271942

2

Synthesis and preliminary pharmacological investigation of new N-substituted-N-[ω-(ω-phenoxy-alkylpiperazin-1-yl)alkyl]guanidines as non-imidazole histamine H(3) antagonists.

Staszewski M, Walczyński K. Staszewski M, et al. Arch Pharm (Weinheim). 2012 Jun;345(6):431-43. doi: 10.1002/ardp.201100428. Epub 2012 Mar 13. Arch Pharm (Weinheim). 2012. PMID: 22415744

3

Non-imidazole histamine H₃ ligands: part V. synthesis and preliminary pharmacological investigation of 1-[2-thiazol-4-yl- and 1-[2-thiazol-5-yl-(2-aminoethyl)]-4-n-propylpiperazine derivatives.

Guryn R, Staszewski M, Walczyński K. Guryn R, et al. Among authors: staszewski m. Med Chem Res. 2013 Aug;22(8):3640-3652. doi: 10.1007/s00044-012-0372-8. Epub 2012 Nov 29. Med Chem Res. 2013. PMID: 23807824 Free PMC article.

4

Loratadine analogues as MAGL inhibitors.

Patel JZ, Ahenkorah S, Vaara M, Staszewski M, Adams Y, Laitinen T, Navia-Paldanius D, Parkkari T, Savinainen JR, Walczyński K, Laitinen JT, Nevalainen TJ. Patel JZ, et al. Among authors: staszewski m. Bioorg Med Chem Lett. 2015 Apr 1;25(7):1436-42. doi: 10.1016/j.bmcl.2015.02.037. Epub 2015 Feb 24. Bioorg Med Chem Lett. 2015. PMID: 25752982

5

Non-Imidazole Histamine H3 Ligands. Part VI. Synthesis and Preliminary Pharmacological Investigation of Thiazole-Type Histamine H3-Receptor Antagonists with Lacking a Nitrogen Nucleus in the Side Chain.

Guryn R, Staszewski M, Kopczacki P, Walczyski K. Guryn R, et al. Among authors: staszewski m. Med Chem. 2016;13(1):65-76. doi: 10.2174/1573406412666160525121158. Med Chem. 2016. PMID: 27220560

6

Non-Imidazole Histamine H₃ Ligands. Part VII. Synthesis, In Vitro and In Vivo Characterization of 5-Substituted-2-thiazol-4-n-propylpiperazines.

Guryn R, Staszewski M, Stasiak A, McNaught Flores D, Fogel WA, Leurs R, Walczyński K. Guryn R, et al. Among authors: staszewski m. Molecules. 2018 Feb 3;23(2):326. doi: 10.3390/molecules23020326. Molecules. 2018. PMID: 29401659 Free PMC article.

7

Design, synthesis, and in vitro and in vivo characterization of 1-{4-[4-(substituted)piperazin-1-yl]butyl}guanidines and their piperidine analogues as histamine H₃ receptor antagonists.

Staszewski M, Stasiak A, Karcz T, McNaught Flores D, Fogel WA, Kieć-Kononowicz K, Leurs R, Walczyński K. Staszewski M, et al. Medchemcomm. 2019 Jan 11;10(2):234-251. doi: 10.1039/c8md00527c. eCollection 2019 Feb 1. Medchemcomm. 2019. PMID: 30881612 Free PMC article.

8

Guanidine Derivatives: How Simple Structural Modification of Histamine H₃R Antagonists Has Led to the Discovery of Potent Muscarinic M₂R/M₄R Antagonists.

Staszewski M, Nelic D, Jończyk J, Dubiel M, Frank A, Stark H, Bajda M, Jakubik J, Walczyński K. Staszewski M, et al. ACS Chem Neurosci. 2021 Jul 7;12(13):2503-2519. doi: 10.1021/acschemneuro.1c00237. Epub 2021 Jun 8. ACS Chem Neurosci. 2021. PMID: 34100603 Free PMC article.

9

Synthesis and Biological Evaluation of Thiazole-Based Derivatives with Potential against Breast Cancer and Antimicrobial Agents.

Pivovarova E, Climova A, Świątkowski M, Staszewski M, Walczyński K, Dzięgielewski M, Bauer M, Kamysz W, Krześlak A, Jóźwiak P, Czylkowska A. Pivovarova E, et al. Among authors: staszewski m. Int J Mol Sci. 2022 Aug 30;23(17):9844. doi: 10.3390/ijms23179844. Int J Mol Sci. 2022. PMID: 36077257 Free PMC article.

10

Guanidines: Synthesis of Novel Histamine H₃R Antagonists with Additional Breast Anticancer Activity and Cholinesterases Inhibitory Effect.

Staszewski M, Iwan M, Werner T, Bajda M, Godyń J, Latacz G, Korga-Plewko A, Kubik J, Szałaj N, Stark H, Malawska B, Więckowska A, Walczyński K. Staszewski M, et al. Pharmaceuticals (Basel). 2023 Apr 30;16(5):675. doi: 10.3390/ph16050675. Pharmaceuticals (Basel). 2023. PMID: 37242458 Free PMC article.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

14 results

Search Page