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C-2 phenyl replacements to obtain potent quinoline-based Staphylococcus aureus NorA inhibitors.
Felicetti T, Mangiaterra G, Cannalire R, Cedraro N, Pietrella D, Astolfi A, Massari S, Tabarrini O, Manfroni G, Barreca ML, Cecchetti V, Biavasco F, Sabatini S. Felicetti T, et al. Among authors: sabatini s. J Enzyme Inhib Med Chem. 2020 Dec;35(1):584-597. doi: 10.1080/14756366.2020.1719083. J Enzyme Inhib Med Chem. 2020. PMID: 31992093 Free PMC article.
Highly potent 1,4-benzothiazine derivatives as K(ATP)-channel openers.
Cecchetti V, Calderone V, Tabarrini O, Sabatini S, Filipponi E, Testai L, Spogli R, Martinotti E, Fravolini A. Cecchetti V, et al. Among authors: sabatini s. J Med Chem. 2003 Aug 14;46(17):3670-9. doi: 10.1021/jm030791q. J Med Chem. 2003. PMID: 12904071
Structure modifications of 6-aminoquinolones with potent anti-HIV activity.
Tabarrini O, Stevens M, Cecchetti V, Sabatini S, Dell'Uomo M, Manfroni G, Palumbo M, Pannecouque C, De Clercq E, Fravolini A. Tabarrini O, et al. Among authors: sabatini s. J Med Chem. 2004 Oct 21;47(22):5567-78. doi: 10.1021/jm049721p. J Med Chem. 2004. PMID: 15481992
429 results