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HCV NS5A replication complex inhibitors. Part 3: discovery of potent analogs with distinct core topologies.
Bioorg Med Chem Lett. 2013 Feb 1;23(3):779-84. doi: 10.1016/j.bmcl.2012.11.086. Epub 2012 Dec 3.
Bioorg Med Chem Lett. 2013.
PMID: 23273521
Synthesis of novel cyclic protease inhibitors using Grubbs olefin metathesis.
Ripka AS, Bohacek RS, Rich DH.
Ripka AS, et al.
Bioorg Med Chem Lett. 1998 Feb 17;8(4):357-60. doi: 10.1016/s0960-894x(98)00025-0.
Bioorg Med Chem Lett. 1998.
PMID: 9871684
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Aspartic protease inhibitors designed from computer-generated templates bind as predicted.
Ripka AS, Satyshur KA, Bohacek RS, Rich DH.
Ripka AS, et al.
Org Lett. 2001 Jul 26;3(15):2309-12. doi: 10.1021/ol016090+.
Org Lett. 2001.
PMID: 11463303
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Peptidomimetic design.
Ripka AS, Rich DH.
Ripka AS, et al.
Curr Opin Chem Biol. 1998 Aug;2(4):441-52. doi: 10.1016/s1367-5931(98)80119-1.
Curr Opin Chem Biol. 1998.
PMID: 9736916
Review.
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First practical synthesis of formamidine ureas and derivatives.
Ripka AS, Díaz DD, Sharpless KB, Finn MG.
Ripka AS, et al.
Org Lett. 2003 May 1;5(9):1531-3. doi: 10.1021/ol034287r.
Org Lett. 2003.
PMID: 12713316
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