Raje MR - Search Results

1

Flex-nucleoside analogues - Novel therapeutics against filoviruses.

Yates MK, Raje MR, Chatterjee P, Spiropoulou CF, Bavari S, Flint M, Soloveva V, Seley-Radtke KL. Yates MK, et al. Among authors: raje mr. Bioorg Med Chem Lett. 2017 Jun 15;27(12):2800-2802. doi: 10.1016/j.bmcl.2017.04.069. Epub 2017 Apr 22. Bioorg Med Chem Lett. 2017. PMID: 28465098 Free PMC article.

2

Synthesis of kojic acid derivatives as secondary binding site probes of D-amino acid oxidase.

Raje M, Hin N, Duvall B, Ferraris DV, Berry JF, Thomas AG, Alt J, Rojas C, Slusher BS, Tsukamoto T. Raje M, et al. Bioorg Med Chem Lett. 2013 Jul 1;23(13):3910-3. doi: 10.1016/j.bmcl.2013.04.062. Epub 2013 May 1. Bioorg Med Chem Lett. 2013. PMID: 23683589 Free PMC article.

3

Discovery of Mcl-1 inhibitors based on a thiazolidine-2,4-dione scaffold.

Whiting E, Raje MR, Chauhan J, Wilder PT, Van Eker D, Hughes SJ, Bowen NG, Vickers GEA, Fenimore IC, Fletcher S. Whiting E, et al. Among authors: raje mr. Bioorg Med Chem Lett. 2018 Feb 1;28(3):523-528. doi: 10.1016/j.bmcl.2017.11.023. Epub 2017 Dec 12. Bioorg Med Chem Lett. 2018. PMID: 29329659

4

Synthetic, structural mimetics of the β-hairpin flap of HIV-1 protease inhibit enzyme function.

Chauhan J, Chen SE, Fenstermacher KJ, Naser-Tavakolian A, Reingewertz T, Salmo R, Lee C, Williams E, Raje M, Sundberg E, DeStefano JJ, Freire E, Fletcher S. Chauhan J, et al. Bioorg Med Chem. 2015 Nov 1;23(21):7095-109. doi: 10.1016/j.bmc.2015.09.002. Epub 2015 Sep 7. Bioorg Med Chem. 2015. PMID: 26474665 Free PMC article.

5

Structure-activity relationship studies and in vivo activity of guanidine-based sphingosine kinase inhibitors: discovery of SphK1- and SphK2-selective inhibitors.

Patwardhan NN, Morris EA, Kharel Y, Raje MR, Gao M, Tomsig JL, Lynch KR, Santos WL. Patwardhan NN, et al. Among authors: raje mr. J Med Chem. 2015 Feb 26;58(4):1879-1899. doi: 10.1021/jm501760d. Epub 2015 Feb 13. J Med Chem. 2015. PMID: 25643074 Free PMC article.

6

Design, synthesis and biological activity of sphingosine kinase 2 selective inhibitors.

Raje MR, Knott K, Kharel Y, Bissel P, Lynch KR, Santos WL. Raje MR, et al. Bioorg Med Chem. 2012 Jan 1;20(1):183-94. doi: 10.1016/j.bmc.2011.11.011. Epub 2011 Nov 15. Bioorg Med Chem. 2012. PMID: 22137932 Free PMC article.

7

Effect of alkyl chain length on sphingosine kinase 2 selectivity.

Knott K, Kharel Y, Raje MR, Lynch KR, Santos WL. Knott K, et al. Among authors: raje mr. Bioorg Med Chem Lett. 2012 Nov 15;22(22):6817-20. doi: 10.1016/j.bmcl.2012.01.050. Epub 2012 Jan 26. Bioorg Med Chem Lett. 2012. PMID: 22321213 Free PMC article.

8

BRD4 Structure-Activity Relationships of Dual PLK1 Kinase/BRD4 Bromodomain Inhibitor BI-2536.

Chen L, Yap JL, Yoshioka M, Lanning ME, Fountain RN, Raje M, Scheenstra JA, Strovel JW, Fletcher S. Chen L, et al. ACS Med Chem Lett. 2015 May 18;6(7):764-9. doi: 10.1021/acsmedchemlett.5b00084. eCollection 2015 Jul 9. ACS Med Chem Lett. 2015. PMID: 26191363 Free PMC article.

9

Towards more drug-like proteomimetics: two-faced, synthetic α-helix mimetics based on a purine scaffold.

Lanning ME, Wilder PT, Bailey H, Drennen B, Cavalier M, Chen L, Yap JL, Raje M, Fletcher S. Lanning ME, et al. Org Biomol Chem. 2015 Aug 28;13(32):8642-6. doi: 10.1039/c5ob00478k. Epub 2015 Jul 24. Org Biomol Chem. 2015. PMID: 26204921 Free PMC article.

10

Molecular mechanisms of 5-HT(3) and NK(1) receptor antagonists in prevention of emesis.

Rojas C, Raje M, Tsukamoto T, Slusher BS. Rojas C, et al. Eur J Pharmacol. 2014 Jan 5;722:26-37. doi: 10.1016/j.ejphar.2013.08.049. Epub 2013 Oct 31. Eur J Pharmacol. 2014. PMID: 24184669 Review.

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