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Contribution of alpha4beta1 integrin to the antiallergic effect of levocabastine.
Biochem Pharmacol. 2008 Sep 15;76(6):751-62. doi: 10.1016/j.bcp.2008.07.007. Epub 2008 Jul 15.
Biochem Pharmacol. 2008.
PMID: 18680729
Nociceptin-induced internalization of the ORL1 receptor in human neuroblastoma cells.
Spampinato S, Di Toro R, Qasem AR.
Spampinato S, et al. Among authors: qasem ar.
Neuroreport. 2001 Oct 8;12(14):3159-63. doi: 10.1097/00001756-200110080-00035.
Neuroreport. 2001.
PMID: 11568656
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Antinociception by a peripherally administered novel endomorphin-1 analogue containing beta-proline.
Spampinato S, Qasem AR, Calienni M, Murari G, Gentilucci L, Tolomelli A, Cardillo G.
Spampinato S, et al. Among authors: qasem ar.
Eur J Pharmacol. 2003 May 23;469(1-3):89-95. doi: 10.1016/s0014-2999(03)01736-9.
Eur J Pharmacol. 2003.
PMID: 12782189
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Endomorphin-1 analogues containing beta-proline are mu-opioid receptor agonists and display enhanced enzymatic hydrolysis resistance.
Cardillo G, Gentilucci L, Qasem AR, Sgarzi F, Spampinato S.
Cardillo G, et al. Among authors: qasem ar.
J Med Chem. 2002 Jun 6;45(12):2571-8. doi: 10.1021/jm011059z.
J Med Chem. 2002.
PMID: 12036366
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Conformational analysis and mu-opioid receptor affinity of short peptides, endomorphin models in a low polarity solvent.
Cardillo G, Gentilucci L, Tolomelli A, Qasem AR, Spampinato S, Calienni M.
Cardillo G, et al. Among authors: qasem ar.
Org Biomol Chem. 2003 Sep 7;1(17):3010-4. doi: 10.1039/b306161m.
Org Biomol Chem. 2003.
PMID: 14518122
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Stability against enzymatic hydrolysis of endomorphin-1 analogues containing beta-proline.
Cardillo G, Gentilucci L, Tolomelli A, Calienni M, Qasem AR, Spampinato S.
Cardillo G, et al. Among authors: qasem ar.
Org Biomol Chem. 2003 May 7;1(9):1498-502. doi: 10.1039/b301507f.
Org Biomol Chem. 2003.
PMID: 12926278
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Synthesis and evaluation of the affinity toward mu-opioid receptors of atypical, lipophilic ligands based on the sequence c[-Tyr-Pro-Trp-Phe-Gly-].
Cardillo G, Gentilucci L, Tolomelli A, Spinosa R, Calienni M, Qasem AR, Spampinato S.
Cardillo G, et al. Among authors: qasem ar.
J Med Chem. 2004 Oct 7;47(21):5198-203. doi: 10.1021/jm0498811.
J Med Chem. 2004.
PMID: 15456262
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Deoxamuscaroneoxime derivatives as useful muscarinic agonists to explore the muscarinic subsite: demox, a modulator of orthosteric and allosteric sites at cardiac muscarinic M2 receptors.
Angeli P, Marucci G, Buccioni M, Piergentili A, Giannella M, Quaglia W, Pigini M, Cantalamessa F, Nasuti C, Novi F, Maggio R, Qasem AR, Spampinato S.
Angeli P, et al. Among authors: qasem ar.
Life Sci. 2002 Feb 8;70(12):1427-46. doi: 10.1016/s0024-3205(01)01521-1.
Life Sci. 2002.
PMID: 11883718
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