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Biological evaluation and spectral characterization of a novel tetracenomycin X congener.
Alferova VA, Maviza TP, Biryukov MV, Zakalyukina YV, Lukianov DA, Skvortsov DA, Vasilyeva LA, Tashlitsky VN, Polshakov VI, Sergiev PV, Korshun VA, Osterman IA. Alferova VA, et al. Among authors: polshakov vi. Biochimie. 2022 Jan;192:63-71. doi: 10.1016/j.biochi.2021.09.014. Epub 2021 Sep 28. Biochimie. 2022. PMID: 34592388
NMR assignments of the WBSCR27 protein related to Williams-Beuren syndrome.
Mariasina SS, Petrova OA, Osterman IA, Sergeeva OV, Efimov SV, Klochkov VV, Sergiev PV, Dontsova OA, Huang TH, Chang CF, Polshakov VI. Mariasina SS, et al. Among authors: polshakov vi. Biomol NMR Assign. 2018 Oct;12(2):303-308. doi: 10.1007/s12104-018-9827-2. Epub 2018 Jun 4. Biomol NMR Assign. 2018. PMID: 29868988
Nybomycin-producing Streptomyces isolated from carpenter ant Camponotus vagus.
Zakalyukina YV, Birykov MV, Lukianov DA, Shiriaev DI, Komarova ES, Skvortsov DA, Kostyukevich Y, Tashlitsky VN, Polshakov VI, Nikolaev E, Sergiev PV, Osterman IA. Zakalyukina YV, et al. Among authors: polshakov vi. Biochimie. 2019 May;160:93-99. doi: 10.1016/j.biochi.2019.02.010. Epub 2019 Feb 21. Biochimie. 2019. PMID: 30797881
Tetracenomycin X inhibits translation by binding within the ribosomal exit tunnel.
Osterman IA, Wieland M, Maviza TP, Lashkevich KA, Lukianov DA, Komarova ES, Zakalyukina YV, Buschauer R, Shiriaev DI, Leyn SA, Zlamal JE, Biryukov MV, Skvortsov DA, Tashlitsky VN, Polshakov VI, Cheng J, Polikanov YS, Bogdanov AA, Osterman AL, Dmitriev SE, Beckmann R, Dontsova OA, Wilson DN, Sergiev PV. Osterman IA, et al. Among authors: polshakov vi. Nat Chem Biol. 2020 Oct;16(10):1071-1077. doi: 10.1038/s41589-020-0578-x. Epub 2020 Jun 29. Nat Chem Biol. 2020. PMID: 32601485
Synthesis and Biological Evaluation of PSMA Ligands with Aromatic Residues and Fluorescent Conjugates Based on Them.
Machulkin AE, Shafikov RR, Uspenskaya AA, Petrov SA, Ber AP, Skvortsov DA, Nimenko EA, Zyk NU, Smirnova GB, Pokrovsky VS, Abakumov MA, Saltykova IV, Akhmirov RT, Garanina AS, Polshakov VI, Saveliev OY, Ivanenkov YA, Aladinskaya AV, Finko AV, Yamansarov EU, Krasnovskaya OO, Erofeev AS, Gorelkin PV, Dontsova OA, Beloglazkina EK, Zyk NV, Khazanova ES, Majouga AG. Machulkin AE, et al. Among authors: polshakov vi. J Med Chem. 2021 Apr 22;64(8):4532-4552. doi: 10.1021/acs.jmedchem.0c01935. Epub 2021 Apr 6. J Med Chem. 2021. PMID: 33822606
Synthesis, Characterization, and Preclinical Evaluation of a Small-Molecule Prostate-Specific Membrane Antigen-Targeted Monomethyl Auristatin E Conjugate.
Machulkin AE, Uspenskaya AA, Zyk NU, Nimenko EA, Ber AP, Petrov SA, Polshakov VI, Shafikov RR, Skvortsov DA, Plotnikova EA, Pankratov AA, Smirnova GB, Borisova YA, Pokrovsky VS, Kolmogorov VS, Vaneev AN, Khudyakov AD, Chepikova OE, Kovalev S, Zamyatnin AA Jr, Erofeev A, Gorelkin P, Beloglazkina EK, Zyk NV, Khazanova ES, Majouga AG. Machulkin AE, et al. Among authors: polshakov vi. J Med Chem. 2021 Dec 9;64(23):17123-17145. doi: 10.1021/acs.jmedchem.1c01157. Epub 2021 Nov 19. J Med Chem. 2021. PMID: 34797052
[Analogs of S-Adenosyl-L-Methionine in Studies of Methyltransferases].
Rudenko AY, Mariasina SS, Sergiev PV, Polshakov VI. Rudenko AY, et al. Among authors: polshakov vi. Mol Biol (Mosk). 2022 Mar-Apr;56(2):296-319. doi: 10.31857/S0026898422020148. Mol Biol (Mosk). 2022. PMID: 35403621 Free article. Review. Russian.
69 results