Neamati N - Search Results

1

Design and synthesis of bis-amide and hydrazide-containing derivatives of malonic acid as potential HIV-1 integrase inhibitors.

Sechi M, Azzena U, Delussu MP, Dallocchio R, Dessì A, Cosseddu A, Pala N, Neamati N. Sechi M, et al. Among authors: neamati n. Molecules. 2008 Oct 1;13(10):2442-61. doi: 10.3390/molecules13102442. Molecules. 2008. PMID: 18830166 Free PMC article.

2

Design and synthesis of novel dihydroxyindole-2-carboxylic acids as HIV-1 integrase inhibitors.

Sechi M, Angotzi G, Dallocchio R, Dessì A, Carta F, Sannia L, Mariani A, Fiori S, Sanchez T, Movsessian L, Plasencia C, Neamati N. Sechi M, et al. Among authors: neamati n. Antivir Chem Chemother. 2004 Mar;15(2):67-81. doi: 10.1177/095632020401500203. Antivir Chem Chemother. 2004. PMID: 15185725 Free article.

3

Design and synthesis of novel indole beta-diketo acid derivatives as HIV-1 integrase inhibitors.

Sechi M, Derudas M, Dallocchio R, Dessì A, Bacchi A, Sannia L, Carta F, Palomba M, Ragab O, Chan C, Shoemaker R, Sei S, Dayam R, Neamati N. Sechi M, et al. Among authors: neamati n. J Med Chem. 2004 Oct 7;47(21):5298-310. doi: 10.1021/jm049944f. J Med Chem. 2004. PMID: 15456274

A plethora of diketo acid-containing compounds have been claimed in patent literature without disclosing much biological activities and synthetic details (reviewed in Neamati, N. Exp. Opin. Ther. Pat. 2002, 12, 709-724). To establish a coherent structure-activity re …

A plethora of diketo acid-containing compounds have been claimed in patent literature without disclosing much biological activities and synt …

4

Design of novel bioisosteres of beta-diketo acid inhibitors of HIV-1 integrase.

Sechi M, Sannia L, Carta F, Palomba M, Dallocchio R, Dessì A, Derudas M, Zawahir Z, Neamati N. Sechi M, et al. Among authors: neamati n. Antivir Chem Chemother. 2005;16(1):41-61. doi: 10.1177/095632020501600105. Antivir Chem Chemother. 2005. PMID: 15739621 Free article.

5

Design and synthesis of novel dihydroquinoline-3-carboxylic acids as HIV-1 integrase inhibitors.

Sechi M, Rizzi G, Bacchi A, Carcelli M, Rogolino D, Pala N, Sanchez TW, Taheri L, Dayam R, Neamati N. Sechi M, et al. Among authors: neamati n. Bioorg Med Chem. 2009 Apr 1;17(7):2925-35. doi: 10.1016/j.bmc.2008.10.088. Epub 2008 Nov 6. Bioorg Med Chem. 2009. PMID: 19026554

6

Design, synthesis, molecular modeling, and anti-HIV-1 integrase activity of a series of photoactivatable diketo acid-containing inhibitors as affinity probes.

Sechi M, Carta F, Sannia L, Dallocchio R, Dessì A, Al-Safi RI, Neamati N. Sechi M, et al. Among authors: neamati n. Antiviral Res. 2009 Mar;81(3):267-76. doi: 10.1016/j.antiviral.2008.12.010. Epub 2009 Jan 9. Antiviral Res. 2009. PMID: 19135482

7

From ligand to complexes: inhibition of human immunodeficiency virus type 1 integrase by beta-diketo acid metal complexes.

Sechi M, Bacchi A, Carcelli M, Compari C, Duce E, Fisicaro E, Rogolino D, Gates P, Derudas M, Al-Mawsawi LQ, Neamati N. Sechi M, et al. Among authors: neamati n. J Med Chem. 2006 Jul 13;49(14):4248-60. doi: 10.1021/jm060193m. J Med Chem. 2006. PMID: 16821784

8

HIV-1 IN strand transfer chelating inhibitors: a focus on metal binding.

Bacchi A, Carcelli M, Compari C, Fisicaro E, Pala N, Rispoli G, Rogolino D, Sanchez TW, Sechi M, Neamati N. Bacchi A, et al. Among authors: neamati n. Mol Pharm. 2011 Apr 4;8(2):507-19. doi: 10.1021/mp100343x. Epub 2011 Mar 8. Mol Pharm. 2011. PMID: 21323359

9

Investigating the role of metal chelation in HIV-1 integrase strand transfer inhibitors.

Bacchi A, Carcelli M, Compari C, Fisicaro E, Pala N, Rispoli G, Rogolino D, Sanchez TW, Sechi M, Sinisi V, Neamati N. Bacchi A, et al. Among authors: neamati n. J Med Chem. 2011 Dec 22;54(24):8407-20. doi: 10.1021/jm200851g. Epub 2011 Nov 22. J Med Chem. 2011. PMID: 22066494

10

Ruthenium arene complexes as HIV-1 integrase strand transfer inhibitors.

Carcelli M, Bacchi A, Pelagatti P, Rispoli G, Rogolino D, Sanchez TW, Sechi M, Neamati N. Carcelli M, et al. Among authors: neamati n. J Inorg Biochem. 2013 Jan;118:74-82. doi: 10.1016/j.jinorgbio.2012.09.021. Epub 2012 Sep 28. J Inorg Biochem. 2013. PMID: 23123342

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