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SAR by Space: Enriching Hit Sets from the Chemical Space.
Klingler FM, Gastreich M, Grygorenko OO, Savych O, Borysko P, Griniukova A, Gubina KE, Lemmen C, Moroz YS. Klingler FM, et al. Among authors: moroz ys. Molecules. 2019 Aug 26;24(17):3096. doi: 10.3390/molecules24173096. Molecules. 2019. PMID: 31454992 Free PMC article.
Facile One-Pot Parallel Synthesis of 3-Amino-1,2,4-triazoles.
Bogolyubsky AV, Savych O, Zhemera AV, Pipko SE, Grishchenko AV, Konovets AI, Doroshchuk RO, Khomenko DN, Brovarets VS, Moroz YS, Vybornyi M. Bogolyubsky AV, et al. Among authors: moroz ys. ACS Comb Sci. 2018 Jul 9;20(7):461-466. doi: 10.1021/acscombsci.8b00060. Epub 2018 Jun 18. ACS Comb Sci. 2018. PMID: 29874036
(Chlorosulfonyl)benzenesulfonyl Fluorides-Versatile Building Blocks for Combinatorial Chemistry: Design, Synthesis and Evaluation of a Covalent Inhibitor Library.
Tolmachova KA, Moroz YS, Konovets A, Platonov MO, Vasylchenko OV, Borysko P, Zozulya S, Gryniukova A, Bogolubsky AV, Pipko S, Mykhailiuk PK, Brovarets VS, Grygorenko OO. Tolmachova KA, et al. Among authors: moroz ys. ACS Comb Sci. 2018 Nov 12;20(11):672-680. doi: 10.1021/acscombsci.8b00130. Epub 2018 Nov 1. ACS Comb Sci. 2018. PMID: 30354064
Evolution of commercially available compounds for HTS.
Volochnyuk DM, Ryabukhin SV, Moroz YS, Savych O, Chuprina A, Horvath D, Zabolotna Y, Varnek A, Judd DB. Volochnyuk DM, et al. Among authors: moroz ys. Drug Discov Today. 2019 Feb;24(2):390-402. doi: 10.1016/j.drudis.2018.10.016. Epub 2018 Nov 3. Drug Discov Today. 2019. PMID: 30399443 Free article. Review.
One-Pot Parallel Synthesis of 5-(Dialkylamino)tetrazoles.
Savych O, Kuchkovska YO, Bogolyubsky AV, Konovets AI, Gubina KE, Pipko SE, Zhemera AV, Grishchenko AV, Khomenko DN, Brovarets VS, Doroschuk R, Moroz YS, Grygorenko OO. Savych O, et al. Among authors: moroz ys. ACS Comb Sci. 2019 Sep 9;21(9):635-642. doi: 10.1021/acscombsci.9b00120. Epub 2019 Aug 29. ACS Comb Sci. 2019. PMID: 31437394 Free PMC article.
85 results