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17β-Hydroxysteroid Dehydrogenase Type 1 Inhibition: A Potential Treatment Option for Non-Small Cell Lung Cancer.
Gargano EM, Mohamed A, Abdelsamie AS, Mangiatordi GF, Drzewiecka H, Jagodziński PP, Mazzini A, van Koppen CJ, Laschke MW, Nicolotti O, Carotti A, Marchais-Oberwinkler S, Hartmann RW, Frotscher M. Gargano EM, et al. Among authors: mangiatordi gf. ACS Med Chem Lett. 2021 Nov 18;12(12):1920-1924. doi: 10.1021/acsmedchemlett.1c00462. eCollection 2021 Dec 9. ACS Med Chem Lett. 2021. PMID: 34917255 Free PMC article.
REACH and in silico methods: an attractive opportunity for medicinal chemists.
Nicolotti O, Benfenati E, Carotti A, Gadaleta D, Gissi A, Mangiatordi GF, Novellino E. Nicolotti O, et al. Among authors: mangiatordi gf. Drug Discov Today. 2014 Nov;19(11):1757-1768. doi: 10.1016/j.drudis.2014.06.027. Epub 2014 Jul 3. Drug Discov Today. 2014. PMID: 24998783 Review.
Trimethoxybenzanilide-based P-glycoprotein modulators: an interesting case of lipophilicity tuning by intramolecular hydrogen bonding.
Tardia P, Stefanachi A, Niso M, Stolfa DA, Mangiatordi GF, Alberga D, Nicolotti O, Lattanzi G, Carotti A, Leonetti F, Perrone R, Berardi F, Azzariti A, Colabufo NA, Cellamare S. Tardia P, et al. Among authors: mangiatordi gf. J Med Chem. 2014 Aug 14;57(15):6403-18. doi: 10.1021/jm500697c. Epub 2014 Aug 5. J Med Chem. 2014. PMID: 25093931
A new gating site in human aquaporin-4: Insights from molecular dynamics simulations.
Alberga D, Nicolotti O, Lattanzi G, Nicchia GP, Frigeri A, Pisani F, Benfenati V, Mangiatordi GF. Alberga D, et al. Among authors: mangiatordi gf. Biochim Biophys Acta. 2014 Dec;1838(12):3052-60. doi: 10.1016/j.bbamem.2014.08.015. Epub 2014 Aug 19. Biochim Biophys Acta. 2014. PMID: 25150048 Free article.
A generalizable definition of chemical similarity for read-across.
Floris M, Manganaro A, Nicolotti O, Medda R, Mangiatordi GF, Benfenati E. Floris M, et al. Among authors: mangiatordi gf. J Cheminform. 2014 Oct 18;6(1):39. doi: 10.1186/s13321-014-0039-1. eCollection 2014 Dec. J Cheminform. 2014. PMID: 25383097 Free PMC article.
88 results