LaPlante SR - Search Results

1

Synthesis and Biological Activity of Hydrazones and Derivatives: A Review.

de Oliveira Carneiro Brum J, França TCC, LaPlante SR, Villar JDF. de Oliveira Carneiro Brum J, et al. Among authors: laplante sr. Mini Rev Med Chem. 2020;20(5):342-368. doi: 10.2174/1389557519666191014142448. Mini Rev Med Chem. 2020. PMID: 31612828 Review.

2

Vinyl fluoride as a mimic of the "intermediate' enol form in the 5 alpha-reductase transformation: synthesis and in vitro activity of (N-1',1'-dimethylethyl)-3-haloandrost-3,5-diene-17 beta-carboxamides.

Li X, Singh SM, Luu-The V, Côté J, Laplante S, Labrie F. Li X, et al. Bioorg Med Chem. 1996 Jan;4(1):55-60. doi: 10.1016/0968-0896(95)00160-3. Bioorg Med Chem. 1996. PMID: 8689240

3

Synthesis of NSC 106084 and NSC 14778 and evaluation of their DNMT inhibitory activity.

Leroy M, Mélin L, LaPlante SR, Medina-Franco JL, Gagnon A. Leroy M, et al. Among authors: laplante sr. Bioorg Med Chem Lett. 2019 Mar 15;29(6):826-831. doi: 10.1016/j.bmcl.2019.01.022. Epub 2019 Jan 22. Bioorg Med Chem Lett. 2019. PMID: 30704813

4

Exposing Small-Molecule Nanoentities by a Nuclear Magnetic Resonance Relaxation Assay.

Ayotte Y, Marando VM, Vaillancourt L, Bouchard P, Heffron G, Coote PW, Larda ST, LaPlante SR. Ayotte Y, et al. Among authors: laplante sr. J Med Chem. 2019 Sep 12;62(17):7885-7896. doi: 10.1021/acs.jmedchem.9b00653. Epub 2019 Sep 3. J Med Chem. 2019. PMID: 31422659

5

Reactivation of VX-Inhibited Human Acetylcholinesterase by Deprotonated Pralidoxime. A Complementary Quantum Mechanical Study.

da Silva JAV, Pereira AF, LaPlante SR, Kuca K, Ramalho TC, França TCC. da Silva JAV, et al. Among authors: laplante sr. Biomolecules. 2020 Jan 27;10(2):192. doi: 10.3390/biom10020192. Biomolecules. 2020. PMID: 32012780 Free PMC article.

6

Synthesis and in vitro evaluation of 4-substituted N-(1,1-dimethylethyl)-3-oxo-4-androstene-17 beta-carboxamides as 5 alpha-reductase inhibitors and antiandrogens.

Li X, Singh SM, Côté J, Laplante S, Veilleux R, Labrie F. Li X, et al. J Med Chem. 1995 Apr 28;38(9):1456-61. doi: 10.1021/jm00009a006. J Med Chem. 1995. PMID: 7739004

7

Synthesis and in vitro study of 17 beta-[N-ureylene-N,N'-disubstituted]-4-methyl-4-aza-5 alpha-androstan-3-ones as selective inhibitors of type I 5 alpha-reductase.

Lourdusamy M, Côté J, Laplante S, Labrie F, Singh SM. Lourdusamy M, et al. Bioorg Med Chem. 1997 Feb;5(2):305-10. doi: 10.1016/s0968-0896(96)00241-6. Bioorg Med Chem. 1997. PMID: 9061195

8

Non-nucleoside inhibitors of the hepatitis C virus NS5B polymerase: discovery and preliminary SAR of benzimidazole derivatives.

Beaulieu PL, Bös M, Bousquet Y, Fazal G, Gauthier J, Gillard J, Goulet S, LaPlante S, Poupart MA, Lefebvre S, McKercher G, Pellerin C, Austel V, Kukolj G. Beaulieu PL, et al. Bioorg Med Chem Lett. 2004 Jan 5;14(1):119-24. doi: 10.1016/j.bmcl.2003.10.023. Bioorg Med Chem Lett. 2004. PMID: 14684311

9

Assessing atropisomer axial chirality in drug discovery and development.

Laplante SR, D Fader L, Fandrick KR, Fandrick DR, Hucke O, Kemper R, Miller SP, Edwards PJ. Laplante SR, et al. J Med Chem. 2011 Oct 27;54(20):7005-22. doi: 10.1021/jm200584g. Epub 2011 Sep 15. J Med Chem. 2011. PMID: 21848318 Review. No abstract available.

10

Identification of benzofurano[3,2-d]pyrimidin-2-ones, a new series of HIV-1 nucleotide-competing reverse transcriptase inhibitors.

Tremblay M, Bethell RC, Cordingley MG, DeRoy P, Duan J, Duplessis M, Edwards PJ, Faucher AM, Halmos T, James CA, Kuhn C, Lacoste JÉ, Lamorte L, LaPlante SR, Malenfant E, Minville J, Morency L, Morin S, Rajotte D, Salois P, Simoneau B, Tremblay S, Sturino CF. Tremblay M, et al. Among authors: laplante sr. Bioorg Med Chem Lett. 2013 May 1;23(9):2775-80. doi: 10.1016/j.bmcl.2013.02.042. Epub 2013 Feb 16. Bioorg Med Chem Lett. 2013. PMID: 23511023

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