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Molecular Mechanism of LEDGF/p75 Dimerization.
Lux V, Brouns T, Čermáková K, Srb P, Fábry M, Mádlíková M, Hořejší M, Kukačka Z, Novák P, Kugler M, Brynda J, DeRijck J, Christ F, Debyser Z, Veverka V. Lux V, et al. Among authors: kugler m. Structure. 2020 Dec 1;28(12):1288-1299.e7. doi: 10.1016/j.str.2020.08.012. Epub 2020 Sep 17. Structure. 2020. PMID: 32946742 Free article.
In situ proteolysis of an N-terminal His tag with thrombin improves the diffraction quality of human aldo-keto reductase 1C3 crystals.
Plavša JJ, Řezáčová P, Kugler M, Pachl P, Brynda J, Voburka Z, Ćelić A, Petri ET, Škerlová J. Plavša JJ, et al. Among authors: kugler m. Acta Crystallogr F Struct Biol Commun. 2018 May 1;74(Pt 5):300-306. doi: 10.1107/S2053230X18005721. Epub 2018 Apr 24. Acta Crystallogr F Struct Biol Commun. 2018. PMID: 29717998 Free PMC article.
Metallacarborane Sulfamides: Unconventional, Specific, and Highly Selective Inhibitors of Carbonic Anhydrase IX.
Grüner B, Brynda J, Das V, Šícha V, Štěpánková J, Nekvinda J, Holub J, Pospíšilová K, Fábry M, Pachl P, Král V, Kugler M, Mašek V, Medvedíková M, Matějková S, Nová A, Lišková B, Gurská S, Džubák P, Hajdúch M, Řezáčová P. Grüner B, et al. Among authors: kugler m. J Med Chem. 2019 Nov 14;62(21):9560-9575. doi: 10.1021/acs.jmedchem.9b00945. Epub 2019 Oct 16. J Med Chem. 2019. PMID: 31568723
Identification of Novel Carbonic Anhydrase IX Inhibitors Using High-Throughput Screening of Pooled Compound Libraries by DNA-Linked Inhibitor Antibody Assay (DIANA).
Tykvart J, Navrátil V, Kugler M, Šácha P, Schimer J, Hlaváčková A, Tenora L, Zemanová J, Dejmek M, Král V, Potáček M, Majer P, Jahn U, Brynda J, Řezáčová P, Konvalinka J. Tykvart J, et al. Among authors: kugler m. SLAS Discov. 2020 Oct;25(9):1026-1037. doi: 10.1177/2472555220918836. Epub 2020 May 26. SLAS Discov. 2020. PMID: 32452709 Free article.
Sulfonamido carboranes as highly selective inhibitors of cancer-specific carbonic anhydrase IX.
Dvořanová J, Kugler M, Holub J, Šícha V, Das V, Nekvinda J, El Anwar S, Havránek M, Pospíšilová K, Fábry M, Král V, Medvedíková M, Matějková S, Lišková B, Gurská S, Džubák P, Brynda J, Hajdúch M, Grüner B, Řezáčová P. Dvořanová J, et al. Among authors: kugler m. Eur J Med Chem. 2020 Aug 15;200:112460. doi: 10.1016/j.ejmech.2020.112460. Epub 2020 May 18. Eur J Med Chem. 2020. PMID: 32505851
Direct Introduction of an Alkylsulfonamido Group on C-sites of Isomeric Dicarba-closo-dodecaboranes: The Influence of Stereochemistry on Inhibitory Activity against the Cancer-Associated Carbonic Anhydrase IX Isoenzyme.
Nekvinda J, Kugler M, Holub J, El Anwar S, Brynda J, Pospíšilová K, Růžičková Z, Řezáčová P, Grüner B. Nekvinda J, et al. Among authors: kugler m. Chemistry. 2020 Dec 9;26(69):16541-16553. doi: 10.1002/chem.202002809. Epub 2020 Nov 3. Chemistry. 2020. PMID: 32757220
106 results