Guillon R - Search Results

1

Highly Selective Phosphatidylinositol 4-Kinase IIIβ Inhibitors and Structural Insight into Their Mode of Action.

Mejdrová I, Chalupská D, Kögler M, Šála M, Plačková P, Baumlová A, Hřebabecký H, Procházková E, Dejmek M, Guillon R, Strunin D, Weber J, Lee G, Birkus G, Mertlíková-Kaiserová H, Boura E, Nencka R. Mejdrová I, et al. Among authors: guillon r. J Med Chem. 2015 May 14;58(9):3767-93. doi: 10.1021/acs.jmedchem.5b00499. Epub 2015 May 4. J Med Chem. 2015. PMID: 25897704

2

Identification of Noncompetitive Inhibitors of Cytosolic 5'-Nucleotidase II Using a Fragment-Based Approach.

Marton Z, Guillon R, Krimm I, Preeti, Rahimova R, Egron D, Jordheim LP, Aghajari N, Dumontet C, Périgaud C, Lionne C, Peyrottes S, Chaloin L. Marton Z, et al. Among authors: guillon r. J Med Chem. 2015 Dec 24;58(24):9680-96. doi: 10.1021/acs.jmedchem.5b01616. Epub 2015 Dec 7. J Med Chem. 2015. PMID: 26599519

3

Lead optimization and biological evaluation of fragment-based cN-II inhibitors.

Guillon R, Rahimova R, Preeti, Egron D, Rouanet S, Dumontet C, Aghajari N, Jordheim LP, Chaloin L, Peyrottes S. Guillon R, et al. Eur J Med Chem. 2019 Apr 15;168:28-44. doi: 10.1016/j.ejmech.2019.02.040. Epub 2019 Feb 14. Eur J Med Chem. 2019. PMID: 30798051

4

New azole antifungals with a fused triazinone scaffold.

Montoir D, Guillon R, Gazzola S, Ourliac-Garnier I, Soklou KE, Tonnerre A, Picot C, Planchat A, Pagniez F, Le Pape P, Logé C. Montoir D, et al. Among authors: guillon r. Eur J Med Chem. 2020 Mar 1;189:112082. doi: 10.1016/j.ejmech.2020.112082. Epub 2020 Jan 20. Eur J Med Chem. 2020. PMID: 32000050

5

Design of new antifungal agents: synthesis and evaluation of 1-[(1H-indol-5-ylmethyl)amino]-2-phenyl-3-(1H-1,2,4-triazol-1-yl)propan-2-ols.

Guillon R, Giraud F, Logé C, Le Borgne M, Picot C, Pagniez F, Le Pape P. Guillon R, et al. Bioorg Med Chem Lett. 2009 Oct 15;19(20):5833-6. doi: 10.1016/j.bmcl.2009.08.089. Epub 2009 Aug 31. Bioorg Med Chem Lett. 2009. PMID: 19762235

6

Synthesis and structure-activity relationships of 2-phenyl-1-[(pyridinyl- and piperidinylmethyl)amino]-3-(1H-1,2,4-triazol-1-yl)propan-2-ols as antifungal agents.

Giraud F, Guillon R, Logé C, Pagniez F, Picot C, Le Borgne M, Le Pape P. Giraud F, et al. Among authors: guillon r. Bioorg Med Chem Lett. 2009 Jan 15;19(2):301-4. doi: 10.1016/j.bmcl.2008.11.101. Epub 2008 Dec 3. Bioorg Med Chem Lett. 2009. PMID: 19091558

7

Synthesis and in vitro antifungal evaluation of 2-(2,4-difluorophenyl)-1-[(1H-indol-3-ylmethyl)methylamino]-3-(1H-1,2,4-triazol-1-yl)propan-2-ols.

Guillon R, Logé C, Pagniez F, Ferchaud-Roucher V, Duflos M, Picot C, Le Pape P. Guillon R, et al. J Enzyme Inhib Med Chem. 2011 Apr;26(2):261-9. doi: 10.3109/14756366.2010.503607. Epub 2010 Aug 9. J Enzyme Inhib Med Chem. 2011. PMID: 20695753

8

Discovery of a novel broad-spectrum antifungal agent derived from albaconazole.

Guillon R, Pagniez F, Picot C, Hédou D, Tonnerre A, Chosson E, Duflos M, Besson T, Logé C, Le Pape P. Guillon R, et al. ACS Med Chem Lett. 2013 Jan 17;4(2):288-92. doi: 10.1021/ml300429p. eCollection 2013 Feb 14. ACS Med Chem Lett. 2013. PMID: 24900660 Free PMC article.

9

Design, synthesis, and in vitro antifungal activity of 1-[(4-substituted-benzyl)methylamino]-2-(2,4-difluorophenyl)-3-(1H-1,2,4-triazol-1-yl)propan-2-ols.

Guillon R, Pagniez F, Giraud F, Crépin D, Picot C, Le Borgne M, Morio F, Duflos M, Logé C, Le Pape P. Guillon R, et al. ChemMedChem. 2011 May 2;6(5):816-25. doi: 10.1002/cmdc.201000530. Epub 2011 Mar 2. ChemMedChem. 2011. PMID: 21370476

10

Design, synthesis, and biological evaluation of 1-[(biarylmethyl)methylamino]-2-(2,4-difluorophenyl)-3-(1H-1,2,4-triazol-1-yl)propan-2-ols as potent antifungal agents: new insights into structure-activity relationships.

Guillon R, Pagniez F, Rambaud C, Picot C, Duflos M, Logé C, Le Pape P. Guillon R, et al. ChemMedChem. 2011 Oct 4;6(10):1806-15. doi: 10.1002/cmdc.201100262. Epub 2011 Jul 11. ChemMedChem. 2011. PMID: 21748853

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