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Development of l-Dopa-containing diketopiperazines as blood-brain barrier shuttle.
Cornacchia C, Marinelli L, Di Rienzo A, Dimmito MP, Serra F, Di Biase G, De Filippis B, Turkez H, Mardinoglu A, Bellezza I, Di Stefano A, Cacciatore I. Cornacchia C, et al. Among authors: di stefano a, di rienzo a, di biase g. Eur J Med Chem. 2022 Dec 5;243:114746. doi: 10.1016/j.ejmech.2022.114746. Epub 2022 Sep 8. Eur J Med Chem. 2022. PMID: 36099749 Free article.
Dimeric L-dopa derivatives as potential prodrugs.
Di Stefano A, Mosciatti B, Cingolani GM, Giorgioni G, Ricciutelli M, Cacciatore I, Sozio P, Claudi F. Di Stefano A, et al. Bioorg Med Chem Lett. 2001 Apr 23;11(8):1085-8. doi: 10.1016/s0960-894x(01)00140-8. Bioorg Med Chem Lett. 2001. PMID: 11327596
Preparation and pharmacological characterization of trans-2-amino-5(6)-fluoro-6(5)-hydroxy-1-phenyl-2,3-dihydro-1H-indenes as D2-like dopamine receptor agonists.
Di Stefano A, Sozio P, Cacciatore I, Cocco A, Giorgioni G, Costa B, Montali M, Lucacchini A, Martini C, Spoto G, Di Pietrantonio F, Di Matteo E, Pinnen F. Di Stefano A, et al. Among authors: di pietrantonio f, di matteo e. J Med Chem. 2005 Apr 7;48(7):2646-54. doi: 10.1021/jm040889k. J Med Chem. 2005. PMID: 15801855
683 results