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2017 1
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2019 5
2020 3
2021 2
2022 3
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Page 1
Novel analgesic/anti-inflammatory agents: 1,5-Diarylpyrrole nitrooxyethyl sulfides and related compounds as Cyclooxygenase-2 inhibitors containing a nitric oxide donor moiety endowed with vasorelaxant properties.
Saletti M, Maramai S, Reale A, Paolino M, Brogi S, Di Capua A, Cappelli A, Giorgi G, D'Avino D, Rossi A, Ghelardini C, Di Cesare Mannelli L, Sardella R, Carotti A, Woelkart G, Klösch B, Bigogno C, Dondio G, Anzini M. Saletti M, et al. Among authors: reale a. Eur J Med Chem. 2022 Nov 5;241:114615. doi: 10.1016/j.ejmech.2022.114615. Epub 2022 Jul 22. Eur J Med Chem. 2022. PMID: 35932568
Design, Synthesis and Characterization of a Visible-Light-Sensitive Molecular Switch and Its PEGylation Towards a Self-Assembling Molecule.
Paolino M, Saletti M, Reale A, Licciardi M, Varvarà P, Marquette A, Léonard J, Bonechi C, Donati A, Giorgi G, Giuliani G, Carlotti B, Ortica F, Latterini L, Gentile M, Paccagnini E, Olivucci M, Cappelli A. Paolino M, et al. Among authors: reale a. Chemistry. 2022 Sep 6;28(50):e202201477. doi: 10.1002/chem.202201477. Epub 2022 Jul 13. Chemistry. 2022. PMID: 35695822 Free PMC article.
Design, synthesis and biological evaluation of 7-substituted 4-phenyl-6H-imidazo[1,5-a]thieno[3,2-f] [1,4]diazepines as safe anxiolytic agents.
Di Capua A, Reale A, Paolino M, Chemi G, Brogi S, Cappelli A, Giorgi G, Grande F, Di Cesare Mannelli L, Ghelardini C, Matucci R, Garofalo A, Anzini M. Di Capua A, et al. Among authors: reale a. Eur J Med Chem. 2020 Aug 15;200:112405. doi: 10.1016/j.ejmech.2020.112405. Epub 2020 May 18. Eur J Med Chem. 2020. PMID: 32492595
Radiosynthesis and Preclinical Evaluation of 11C-VA426, a Cyclooxygenase-2 Selective Ligand.
Carpinelli A, Rainone P, Belloli S, Reale A, Cappelli A, Germano G, Murtaj V, Coliva A, Di Grigoli G, Valeri A, Gilardi MC, Gianolli L, Anzini M, Moresco RM. Carpinelli A, et al. Among authors: reale a. Contrast Media Mol Imaging. 2019 Sep 24;2019:5823261. doi: 10.1155/2019/5823261. eCollection 2019. Contrast Media Mol Imaging. 2019. PMID: 31598112 Free PMC article.
Physicochemical Properties of A New PEGylated Polybenzofulvene Brush for Drug Encapsulation.
Paolino M, Reale A, Razzano V, Giuliani G, Donati A, Giorgi G, Boccia AC, Mendichi R, Piovani D, Botta C, Salvini L, Samperi F, Savoca C, Licciardi M, Paccagnini E, Gentile M, Cappelli A. Paolino M, et al. Among authors: reale a. Pharmaceutics. 2019 Sep 1;11(9):444. doi: 10.3390/pharmaceutics11090444. Pharmaceutics. 2019. PMID: 31480633 Free PMC article.
Synthesis, biological evaluation and molecular modeling of novel selective COX-2 inhibitors: sulfide, sulfoxide, and sulfone derivatives of 1,5-diarylpyrrol-3-substituted scaffold.
Reale A, Brogi S, Chelini A, Paolino M, Di Capua A, Giuliani G, Cappelli A, Giorgi G, Chemi G, Grillo A, Valoti M, Sautebin L, Rossi A, Pace S, La Motta C, Di Cesare Mannelli L, Lucarini E, Ghelardini C, Anzini M. Reale A, et al. Bioorg Med Chem. 2019 Oct 1;27(19):115045. doi: 10.1016/j.bmc.2019.115045. Epub 2019 Aug 9. Bioorg Med Chem. 2019. PMID: 31427145
17 results