The novel potent TEAD inhibitor, K-975, inhibits YAP1/TAZ-TEAD protein-protein interactions and exerts an anti-tumor effect on malignant pleural mesothelioma.
Kaneda A, Seike T, Danjo T, Nakajima T, Otsubo N, Yamaguchi D, Tsuji Y, Hamaguchi K, Yasunaga M, Nishiya Y, Suzuki M, Saito JI, Yatsunami R, Nakamura S, Sekido Y, Mori K.
Kaneda A, et al. Among authors: yatsunami r.
Am J Cancer Res. 2020 Dec 1;10(12):4399-4415. eCollection 2020.
Am J Cancer Res. 2020.
PMID: 33415007
Free PMC article.