Schirmeister T - Search Results

1

Identification, Characterization, and Synthesis of Natural Parasitic Cysteine Protease Inhibitors: Pentacitidins Are More Potent Falcitidin Analogues.

Brinkmann S, Semmler S, Kersten C, Patras MA, Kurz M, Fuchs N, Hammerschmidt SJ, Legac J, Hammann PE, Vilcinskas A, Rosenthal PJ, Schirmeister T, Bauer A, Schäberle TF. Brinkmann S, et al. Among authors: schirmeister t. ACS Chem Biol. 2022 Mar 18;17(3):576-589. doi: 10.1021/acschembio.1c00861. Epub 2022 Mar 9. ACS Chem Biol. 2022. PMID: 35262340

2

Screening of protease inhibitors as antiplasmodial agents. Part I: Aziridines and epoxides.

Schulz F, Gelhaus C, Degel B, Vicik R, Heppner S, Breuning A, Leippe M, Gut J, Rosenthal PJ, Schirmeister T. Schulz F, et al. Among authors: schirmeister t. ChemMedChem. 2007 Aug;2(8):1214-24. doi: 10.1002/cmdc.200700070. ChemMedChem. 2007. PMID: 17562535

3

Synthesis and evaluation of non-peptidic cysteine protease inhibitors of P. falciparum derived from etacrynic acid.

Dude MA, Kaeppler U, Herb M, Schiller M, Schulz F, Vedder B, Heppner S, Pradel G, Gut J, Rosenthal PJ, Schirmeister T, Leippe M, Gelhaus C. Dude MA, et al. Among authors: schirmeister t. Molecules. 2008 Dec 23;14(1):19-35. doi: 10.3390/molecules14010019. Molecules. 2008. PMID: 19104483 Free PMC article.

4

On-bead screening of a combinatorial fumaric acid derived peptide library yields antiplasmodial cysteine protease inhibitors with unusual peptide sequences.

Machon U, Büchold C, Stempka M, Schirmeister T, Gelhaus C, Leippe M, Gut J, Rosenthal PJ, Kisker C, Leyh M, Schmuck C. Machon U, et al. Among authors: schirmeister t. J Med Chem. 2009 Sep 24;52(18):5662-72. doi: 10.1021/jm900629w. J Med Chem. 2009. PMID: 19715342

5

Michael acceptor based antiplasmodial and antitrypanosomal cysteine protease inhibitors with unusual amino acids.

Breuning A, Degel B, Schulz F, Büchold C, Stempka M, Machon U, Heppner S, Gelhaus C, Leippe M, Leyh M, Kisker C, Rath J, Stich A, Gut J, Rosenthal PJ, Schmuck C, Schirmeister T. Breuning A, et al. Among authors: schirmeister t. J Med Chem. 2010 Mar 11;53(5):1951-63. doi: 10.1021/jm900946n. J Med Chem. 2010. PMID: 20131843

6

New cis-configured aziridine-2-carboxylates as aspartic acid protease inhibitors.

Büchold C, Hemberger Y, Heindl C, Welker A, Degel B, Pfeuffer T, Staib P, Schneider S, Rosenthal PJ, Gut J, Morschhäuser J, Bringmann G, Schirmeister T. Büchold C, et al. Among authors: schirmeister t. ChemMedChem. 2011 Jan 3;6(1):141-52. doi: 10.1002/cmdc.201000370. ChemMedChem. 2011. PMID: 21082722

7

Development of antitrypanosomal and antiplasmodial nonpeptidic cysteine protease inhibitors based on N-protected-guanidino-furan and -pyrrole building blocks.

Langolf S, Machon U, Ehlers M, Sicking W, Schirmeister T, Büchhold C, Gelhaus C, Rosenthal PJ, Schmuck C. Langolf S, et al. Among authors: schirmeister t. ChemMedChem. 2011 Sep 5;6(9):1581-6. doi: 10.1002/cmdc.201100189. Epub 2011 Jun 15. ChemMedChem. 2011. PMID: 21678556 No abstract available.

8

Development of Novel Peptide-Based Michael Acceptors Targeting Rhodesain and Falcipain-2 for the Treatment of Neglected Tropical Diseases (NTDs).

Previti S, Ettari R, Cosconati S, Amendola G, Chouchene K, Wagner A, Hellmich UA, Ulrich K, Krauth-Siegel RL, Wich PR, Schmid I, Schirmeister T, Gut J, Rosenthal PJ, Grasso S, Zappalà M. Previti S, et al. Among authors: schirmeister t. J Med Chem. 2017 Aug 24;60(16):6911-6923. doi: 10.1021/acs.jmedchem.7b00405. Epub 2017 Aug 11. J Med Chem. 2017. PMID: 28763614

9

New aziridine-based inhibitors of cathepsin L-like cysteine proteases with selectivity for the Leishmania cysteine protease LmCPB2.8.

Fey P, Chartomatsidou R, Kiefer W, Mottram JC, Kersten C, Schirmeister T. Fey P, et al. Among authors: schirmeister t. Eur J Med Chem. 2018 Aug 5;156:587-597. doi: 10.1016/j.ejmech.2018.07.012. Epub 2018 Jul 9. Eur J Med Chem. 2018. PMID: 30029081

10

Cis autocatalytic cleavage of glycine-linked Zika virus NS2B-NS3 protease constructs.

von Hammerstein F, Lauth LM, Hammerschmidt S, Wagner A, Schirmeister T, Hellmich UA. von Hammerstein F, et al. Among authors: schirmeister t. FEBS Lett. 2019 Aug;593(16):2204-2213. doi: 10.1002/1873-3468.13507. Epub 2019 Jul 9. FEBS Lett. 2019. PMID: 31240714 Free article.

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