Nieto FR - Search Results

1

Chemoenzymatic synthesis of 2,6-disubstituted tetrahydropyrans with high σ₁ receptor affinity, antitumor and analgesic activity.

Kopp N, Civenni G, Marson D, Laurini E, Pricl S, Catapano CV, Humpf HU, Almansa C, Nieto FR, Schepmann D, Wünsch B. Kopp N, et al. Among authors: nieto fr. Eur J Med Chem. 2021 Jul 5;219:113443. doi: 10.1016/j.ejmech.2021.113443. Epub 2021 Apr 20. Eur J Med Chem. 2021. PMID: 33901806

2

Synthesis, Receptor Affinity, and Antiallodynic Activity of Spirocyclic σ Receptor Ligands with Exocyclic Amino Moiety.

Bergkemper M, Kronenberg E, Thum S, Börgel F, Daniliuc C, Schepmann D, Nieto FR, Brust P, Reinoso RF, Alvarez I, Wünsch B. Bergkemper M, et al. Among authors: nieto fr. J Med Chem. 2018 Nov 8;61(21):9666-9690. doi: 10.1021/acs.jmedchem.8b01183. Epub 2018 Oct 24. J Med Chem. 2018. PMID: 30350997

3

Tetrahydro-3-benzazepines with fluorinated side chains as NMDA and σ₁ receptor antagonists: Synthesis, receptor affinity, selectivity and antiallodynic activity.

Thum S, Schepmann D, Ayet E, Pujol M, Nieto FR, Ametamey SM, Wünsch B. Thum S, et al. Among authors: nieto fr. Eur J Med Chem. 2019 Sep 1;177:47-62. doi: 10.1016/j.ejmech.2019.05.034. Epub 2019 May 16. Eur J Med Chem. 2019. PMID: 31129453

4

Discovery of a σ₁ receptor antagonist by combination of unbiased cell painting and thermal proteome profiling.

Wilke J, Kawamura T, Xu H, Brause A, Friese A, Metz M, Schepmann D, Wünsch B, Artacho-Cordón A, Nieto FR, Watanabe N, Osada H, Ziegler S, Waldmann H. Wilke J, et al. Among authors: nieto fr. Cell Chem Biol. 2021 Jun 17;28(6):848-854.e5. doi: 10.1016/j.chembiol.2021.01.009. Epub 2021 Feb 9. Cell Chem Biol. 2021. PMID: 33567254 Free article.

5

Synthesis of tropane-based σ₁ receptor antagonists with antiallodynic activity.

Bechthold E, Schreiber JA, Ritter N, Grey L, Schepmann D, Daniliuc C, González-Cano R, Nieto FR, Seebohm G, Wünsch B. Bechthold E, et al. Among authors: nieto fr. Eur J Med Chem. 2022 Feb 15;230:114113. doi: 10.1016/j.ejmech.2022.114113. Epub 2022 Jan 13. Eur J Med Chem. 2022. PMID: 35065412

6

Conformationally Restricted σ₁ Receptor Antagonists from (-)-Isopulegol.

Blicker L, González-Cano R, Laurini E, Nieto FR, Schmidt J, Schepmann D, Pricl S, Wünsch B. Blicker L, et al. Among authors: nieto fr. J Med Chem. 2023 Apr 13;66(7):4999-5020. doi: 10.1021/acs.jmedchem.2c02081. Epub 2023 Mar 22. J Med Chem. 2023. PMID: 36946301 Free article.

7

Potentiation of morphine-induced mechanical antinociception by σ₁ receptor inhibition: role of peripheral σ₁ receptors.

Sánchez-Fernández C, Nieto FR, González-Cano R, Artacho-Cordón A, Romero L, Montilla-García Á, Zamanillo D, Baeyens JM, Entrena JM, Cobos EJ. Sánchez-Fernández C, et al. Among authors: nieto fr. Neuropharmacology. 2013 Jul;70:348-58. doi: 10.1016/j.neuropharm.2013.03.002. Epub 2013 Mar 21. Neuropharmacology. 2013. PMID: 23524304

8

Antiallodynic and analgesic effects of maslinic acid, a pentacyclic triterpenoid from Olea europaea.

Nieto FR, Cobos EJ, Entrena JM, Parra A, García-Granados A, Baeyens JM. Nieto FR, et al. J Nat Prod. 2013 Apr 26;76(4):737-40. doi: 10.1021/np300783a. Epub 2013 Mar 29. J Nat Prod. 2013. PMID: 23540838

9

Targeting immune-driven opioid analgesia by sigma-1 receptors: Opening the door to novel perspectives for the analgesic use of sigma-1 antagonists.

Tejada MÁ, Montilla-García Á, González-Cano R, Bravo-Caparrós I, Ruiz-Cantero MC, Nieto FR, Cobos EJ. Tejada MÁ, et al. Among authors: nieto fr. Pharmacol Res. 2018 May;131:224-230. doi: 10.1016/j.phrs.2018.02.008. Epub 2018 Feb 15. Pharmacol Res. 2018. PMID: 29454675 Free article. Review.

10

Antagonism by haloperidol and its metabolites of mechanical hypersensitivity induced by intraplantar capsaicin in mice: role of sigma-1 receptors.

Entrena JM, Cobos EJ, Nieto FR, Cendán CM, Baeyens JM, Del Pozo E. Entrena JM, et al. Among authors: nieto fr. Psychopharmacology (Berl). 2009 Jul;205(1):21-33. doi: 10.1007/s00213-009-1513-8. Epub 2009 Mar 27. Psychopharmacology (Berl). 2009. PMID: 19326101 Free PMC article.

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