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Steered Molecular Dynamics Simulations Study on FABP4 Inhibitors.
Tomarchio R, Patamia V, Zagni C, Crocetti L, Cilibrizzi A, Floresta G, Rescifina A. Tomarchio R, et al. Among authors: cilibrizzi a. Molecules. 2023 Mar 17;28(6):2731. doi: 10.3390/molecules28062731. Molecules. 2023. PMID: 36985701 Free PMC article.
Functionalized pyrazoles and pyrazolo[3,4-d]pyridazinones: Synthesis and evaluation of their phosphodiesterase 4 inhibitory activity.
Biagini P, Biancalani C, Graziano A, Cesari N, Giovannoni MP, Cilibrizzi A, Dal Piaz V, Vergelli C, Crocetti L, Delcanale M, Armani E, Rizzi A, Puccini P, Gallo PM, Spinabelli D, Caruso P. Biagini P, et al. Among authors: cilibrizzi a. Bioorg Med Chem. 2010 May 15;18(10):3506-17. doi: 10.1016/j.bmc.2010.03.066. Epub 2010 Mar 31. Bioorg Med Chem. 2010. PMID: 20413313
Further studies on 2-arylacetamide pyridazin-3(2H)-ones: design, synthesis and evaluation of 4,6-disubstituted analogs as formyl peptide receptors (FPRs) agonists.
Giovannoni MP, Schepetkin IA, Cilibrizzi A, Crocetti L, Khlebnikov AI, Dahlgren C, Graziano A, Dal Piaz V, Kirpotina LN, Zerbinati S, Vergelli C, Quinn MT. Giovannoni MP, et al. Among authors: cilibrizzi a. Eur J Med Chem. 2013 Jun;64:512-28. doi: 10.1016/j.ejmech.2013.03.066. Epub 2013 Apr 8. Eur J Med Chem. 2013. PMID: 23685570 Free PMC article.
Further studies on pyrazolo[1',5':1,6]pyrimido[4,5-d]pyridazin-4(3H)-ones as potent and selective human A1 adenosine receptor antagonists.
Giovannoni MP, Ciciani G, Cilibrizzi A, Crocetti L, Daniele S, Di Cesare Mannelli L, Ghelardini C, Giacomelli C, Guerrini G, Martini C, Trincavelli ML, Vergelli C. Giovannoni MP, et al. Among authors: cilibrizzi a. Eur J Med Chem. 2015 Jan 7;89:32-41. doi: 10.1016/j.ejmech.2014.10.020. Epub 2014 Oct 12. Eur J Med Chem. 2015. PMID: 25462223
Cinnoline derivatives as human neutrophil elastase inhibitors.
Giovannoni MP, Schepetkin IA, Crocetti L, Ciciani G, Cilibrizzi A, Guerrini G, Khlebnikov AI, Quinn MT, Vergelli C. Giovannoni MP, et al. Among authors: cilibrizzi a. J Enzyme Inhib Med Chem. 2016 Aug;31(4):628-39. doi: 10.3109/14756366.2015.1057718. Epub 2015 Jul 21. J Enzyme Inhib Med Chem. 2016. PMID: 26194018 Free PMC article.
58 results