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Page 1
Novel Copper-Containing Cytotoxic Agents Based on 2-Thioxoimidazolones.
Krasnovskaya OO, Guk DA, Naumov AE, Nikitina VN, Semkina AS, Vlasova KY, Pokrovsky V, Ryabaya OO, Karshieva SS, Skvortsov DA, Zhirkina IV, Shafikov RR, Gorelkin PV, Vaneev AN, Erofeev AS, Mazur DM, Tafeenko VA, Pergushov VI, Melnikov MY, Soldatov MA, Shapovalov VV, Soldatov AV, Akasov RA, Gerasimov VM, Sakharov DA, Moiseeva AA, Zyk NV, Beloglazkina EK, Majouga AG. Krasnovskaya OO, et al. Among authors: beloglazkina ek. J Med Chem. 2020 Nov 12;63(21):13031-13063. doi: 10.1021/acs.jmedchem.0c01196. Epub 2020 Oct 20. J Med Chem. 2020. PMID: 32985193
Cleavage of the C-S bond with the formation of a binuclear copper complex with 2-thiolato-3-phenyl-5-(pyridine-2-ylmethylene)-3,5-dihydro-4H-imidazole-4-one. A new mimic of the active site of N2O reductase.
Majouga AG, Beloglazkina EK, Moiseeva AA, Shilova OV, Manzheliy EA, Lebedeva MA, Davies ES, Khlobystov AN, Zyk NV. Majouga AG, et al. Among authors: beloglazkina ek. Dalton Trans. 2013 May 14;42(18):6290-3. doi: 10.1039/c3dt50422k. Dalton Trans. 2013. PMID: 23525195
Mixed valence copper(I,II) binuclear complexes with unexpected structure: synthesis, biological properties and anticancer activity.
Majouga AG, Zvereva MI, Rubtsova MP, Skvortsov DA, Mironov AV, Azhibek DM, Krasnovskaya OO, Gerasimov VM, Udina AV, Vorozhtsov NI, Beloglazkina EK, Agron L, Mikhina LV, Tretyakova AV, Zyk NV, Zefirov NS, Kabanov AV, Dontsova OA. Majouga AG, et al. Among authors: beloglazkina ek. J Med Chem. 2014 Jul 24;57(14):6252-8. doi: 10.1021/jm500154f. Epub 2014 Jul 8. J Med Chem. 2014. PMID: 24950478
Enzyme-functionalized gold-coated magnetite nanoparticles as novel hybrid nanomaterials: synthesis, purification and control of enzyme function by low-frequency magnetic field.
Majouga A, Sokolsky-Papkov M, Kuznetsov A, Lebedev D, Efremova M, Beloglazkina E, Rudakovskaya P, Veselov M, Zyk N, Golovin Y, Klyachko N, Kabanov A. Majouga A, et al. Colloids Surf B Biointerfaces. 2015 Jan 1;125:104-9. doi: 10.1016/j.colsurfb.2014.11.012. Epub 2014 Nov 20. Colloids Surf B Biointerfaces. 2015. PMID: 25460600
Design, synthesis and biological evaluation of novel potent MDM2/p53 small-molecule inhibitors.
Ivanenkov YA, Vasilevski SV, Beloglazkina EK, Kukushkin ME, Machulkin AE, Veselov MS, Chufarova NV, Chernyaginab ES, Vanzcool AS, Zyk NV, Skvortsov DA, Khutornenko AA, Rusanov AL, Tonevitsky AG, Dontsova OA, Majouga AG. Ivanenkov YA, et al. Among authors: beloglazkina ek. Bioorg Med Chem Lett. 2015 Jan 15;25(2):404-9. doi: 10.1016/j.bmcl.2014.09.070. Epub 2014 Oct 2. Bioorg Med Chem Lett. 2015. PMID: 25479770
Synthesis, isomerization and biological activity of novel 2-selenohydantoin derivatives.
Ivanenkov YA, Veselov MS, Rezekin IG, Skvortsov DA, Sandulenko YB, Polyakova MV, Bezrukov DS, Vasilevsky SV, Kukushkin ME, Moiseeva AA, Finko AV, Koteliansky VE, Klyachko NL, Filatova LA, Beloglazkina EK, Zyk NV, Majouga AG. Ivanenkov YA, et al. Among authors: beloglazkina ek. Bioorg Med Chem. 2016 Feb 15;24(4):802-11. doi: 10.1016/j.bmc.2015.12.050. Epub 2016 Jan 2. Bioorg Med Chem. 2016. PMID: 26780833
Small-molecule PSMA ligands. Current state, SAR and perspectives.
Machulkin AE, Ivanenkov YA, Aladinskaya AV, Veselov MS, Aladinskiy VA, Beloglazkina EK, Koteliansky VE, Shakhbazyan AG, Sandulenko YB, Majouga AG. Machulkin AE, et al. Among authors: beloglazkina ek. J Drug Target. 2016 Sep;24(8):679-93. doi: 10.3109/1061186X.2016.1154564. Epub 2016 Mar 10. J Drug Target. 2016. PMID: 26887438 Review.
Identification of Novel Small-Molecule ASGP-R Ligands.
Majouga AG, Ivanenkov YA, Veselov MS, Lopuhov AV, Maklakova SV, Beloglazkina EK, Binevski PV, Klyachko NL, Sandulenko YB, Galkina NY, Koteliansky VE. Majouga AG, et al. Among authors: beloglazkina ek. Curr Drug Deliv. 2016;13(8):1303-1312. doi: 10.2174/1567201813666160719144651. Curr Drug Deliv. 2016. PMID: 27440073
New copper(II) thiohydantoin complexes: Synthesis, characterization, and assessment of their interaction with bovine serum albumin and DNA.
Tishchenko K, Beloglazkina E, Proskurnin M, Malinnikov V, Guk D, Muratova M, Krasnovskaya O, Udina A, Skvortsov D, Shafikov RR, Ivanenkov Y, Aladinskiy V, Sorokin I, Gromov O, Majouga A, Zyk N. Tishchenko K, et al. J Inorg Biochem. 2017 Oct;175:190-197. doi: 10.1016/j.jinorgbio.2017.07.015. Epub 2017 Jul 21. J Inorg Biochem. 2017. PMID: 28756175
68 results