Almansa C - Search Results

1

Chemoenzymatic synthesis of 2,6-disubstituted tetrahydropyrans with high σ₁ receptor affinity, antitumor and analgesic activity.

Kopp N, Civenni G, Marson D, Laurini E, Pricl S, Catapano CV, Humpf HU, Almansa C, Nieto FR, Schepmann D, Wünsch B. Kopp N, et al. Among authors: almansa c. Eur J Med Chem. 2021 Jul 5;219:113443. doi: 10.1016/j.ejmech.2021.113443. Epub 2021 Apr 20. Eur J Med Chem. 2021. PMID: 33901806

2

Synthesis and structure-activity relationships of 1-acyl-4-((2-methyl-3-pyridyl)cyanomethyl)piperazines as PAF antagonists.

Carceller E, Merlos M, Giral M, Almansa C, Bartrolí J, García-Rafanell J, Forn J. Carceller E, et al. Among authors: almansa c. J Med Chem. 1993 Oct 1;36(20):2984-97. doi: 10.1021/jm00072a019. J Med Chem. 1993. PMID: 8411016

3

Synthesis and structure-activity relationship of a new series of potent AT1 selective angiotensin II receptor antagonists: 5-(biphenyl-4-ylmethyl)pyrazoles.

Almansa C, Gómez LA, Cavalcanti FL, de Arriba AF, García-Rafanell J, Forn J. Almansa C, et al. J Med Chem. 1997 Feb 14;40(4):547-58. doi: 10.1021/jm9604383. J Med Chem. 1997. PMID: 9046346

4

Synthesis and SAR of a new series of COX-2-selective inhibitors: pyrazolo[1,5-a]pyrimidines.

Almansa C, de Arriba AF, Cavalcanti FL, Gómez LA, Miralles A, Merlos M, García-Rafanell J, Forn J. Almansa C, et al. J Med Chem. 2001 Feb 1;44(3):350-61. doi: 10.1021/jm0009383. J Med Chem. 2001. PMID: 11462976

5

Synthesis and biological evaluation of the 1-arylpyrazole class of σ(1) receptor antagonists: identification of 4-{2-[5-methyl-1-(naphthalen-2-yl)-1H-pyrazol-3-yloxy]ethyl}morpholine (S1RA, E-52862).

Díaz JL, Cuberes R, Berrocal J, Contijoch M, Christmann U, Fernández A, Port A, Holenz J, Buschmann H, Laggner C, Serafini MT, Burgueño J, Zamanillo D, Merlos M, Vela JM, Almansa C. Díaz JL, et al. Among authors: almansa c. J Med Chem. 2012 Oct 11;55(19):8211-24. doi: 10.1021/jm3007323. Epub 2012 Jul 27. J Med Chem. 2012. PMID: 22784008

6

Synthesis and biological evaluation of a new series of hexahydro-2H-pyrano[3,2-c]quinolines as novel selective σ1 receptor ligands.

Díaz JL, Christmann U, Fernández A, Luengo M, Bordas M, Enrech R, Carro M, Pascual R, Burgueño J, Merlos M, Benet-Buchholz J, Cerón-Bertran J, Ramírez J, Reinoso RF, Fernández de Henestrosa AR, Vela JM, Almansa C. Díaz JL, et al. Among authors: almansa c. J Med Chem. 2013 May 9;56(9):3656-65. doi: 10.1021/jm400181k. Epub 2013 Apr 26. J Med Chem. 2013. PMID: 23560650

7

Selective sigma-1 receptor antagonists for the treatment of pain.

Almansa C, Vela JM. Almansa C, et al. Future Med Chem. 2014 Jun;6(10):1179-99. doi: 10.4155/fmc.14.54. Future Med Chem. 2014. PMID: 25078137 Review.

8

Synthesis and structure-activity relationship study of a new series of selective σ(1) receptor ligands for the treatment of pain: 4-aminotriazoles.

Díaz JL, Christmann U, Fernández A, Torrens A, Port A, Pascual R, Álvarez I, Burgueño J, Monroy X, Montero A, Balada A, Vela JM, Almansa C. Díaz JL, et al. Among authors: almansa c. J Med Chem. 2015 Mar 12;58(5):2441-51. doi: 10.1021/jm501920g. Epub 2015 Feb 19. J Med Chem. 2015. PMID: 25658964

9

Synthesis and Structure-Affinity Relationships of Spirocyclic Benzopyrans with Exocyclic Amino Moiety.

Kronenberg E, Weber F, Brune S, Schepmann D, Almansa C, Friedland K, Laurini E, Pricl S, Wünsch B. Kronenberg E, et al. Among authors: almansa c. J Med Chem. 2019 Apr 25;62(8):4204-4217. doi: 10.1021/acs.jmedchem.9b00449. Epub 2019 Apr 12. J Med Chem. 2019. PMID: 30939014 Free article.

10

Pharmacological characterization of high-affinity σ₁ receptor ligands with spirocyclic thienopyran and thienofuran scaffold.

Schepmann D, Neue C, Westphälinger S, Müller C, Bracher F, Lange C, Bednarski P, Almansa C, Friedland K, Räbiger V, Düfer M, Wünsch B. Schepmann D, et al. Among authors: almansa c. J Pharm Pharmacol. 2020 Feb;72(2):236-248. doi: 10.1111/jphp.13196. Epub 2019 Nov 19. J Pharm Pharmacol. 2020. PMID: 31743446

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