Reilly SW - Search Results

1

A Chemical Approach for Programmable Protein Outputs Based on Engineered Cell Interactions.

Jacome DA, Northrup JD, Ruff AJ, Reilly SW, Lee IK, Blizard GS, Sellmyer MA. Jacome DA, et al. Among authors: reilly sw. ACS Chem Biol. 2021 Jan 15;16(1):52-57. doi: 10.1021/acschembio.0c00935. Epub 2020 Dec 22. ACS Chem Biol. 2021. PMID: 33351606 Free PMC article.

2

Highly Selective Dopamine D₃ Receptor Antagonists with Arylated Diazaspiro Alkane Cores.

Reilly SW, Griffin S, Taylor M, Sahlholm K, Weng CC, Xu K, Jacome DA, Luedtke RR, Mach RH. Reilly SW, et al. J Med Chem. 2017 Dec 14;60(23):9905-9910. doi: 10.1021/acs.jmedchem.7b01248. Epub 2017 Nov 21. J Med Chem. 2017. PMID: 29125762 Free PMC article.

3

Leveraging a Low-Affinity Diazaspiro Orthosteric Fragment to Reduce Dopamine D₃ Receptor (D₃R) Ligand Promiscuity across Highly Conserved Aminergic G-Protein-Coupled Receptors (GPCRs).

Reilly SW, Riad AA, Hsieh CJ, Sahlholm K, Jacome DA, Griffin S, Taylor M, Weng CC, Xu K, Kirschner N, Luedtke RR, Parry C, Malhotra S, Karanicolas J, Mach RH. Reilly SW, et al. J Med Chem. 2019 May 23;62(10):5132-5147. doi: 10.1021/acs.jmedchem.9b00412. Epub 2019 May 6. J Med Chem. 2019. PMID: 31021617

4

Altering Nitrogen Heterocycles of AZD2461 Affords High Affinity Poly(ADP-ribose) Polymerase-1 Inhibitors with Decreased P-Glycoprotein Interactions.

Reilly SW, Puentes LN, Hsieh CJ, Makvandi M, Mach RH. Reilly SW, et al. ACS Omega. 2018 Aug 31;3(8):9997-10001. doi: 10.1021/acsomega.8b00896. Epub 2018 Aug 28. ACS Omega. 2018. PMID: 30198004 Free PMC article.

5

Ligand with Two Modes of Interaction with the Dopamine D₂ Receptor-An Induced-Fit Mechanism of Insurmountable Antagonism.

Ågren R, Zeberg H, Stępniewski TM, Free RB, Reilly SW, Luedtke RR, Århem P, Ciruela F, Sibley DR, Mach RH, Selent J, Nilsson J, Sahlholm K. Ågren R, et al. Among authors: reilly sw. ACS Chem Neurosci. 2020 Oct 7;11(19):3130-3143. doi: 10.1021/acschemneuro.0c00477. Epub 2020 Sep 15. ACS Chem Neurosci. 2020. PMID: 32865974 Free PMC article.

6

Late-Stage Carbon Isotope Exchange of Aryl Nitriles through Ni-Catalyzed C-CN Bond Activation.

Reilly SW, Lam YH, Ren S, Strotman NA. Reilly SW, et al. J Am Chem Soc. 2021 Mar 31;143(12):4817-4823. doi: 10.1021/jacs.1c01454. Epub 2021 Mar 16. J Am Chem Soc. 2021. PMID: 33725443

7

Examination of Diazaspiro Cores as Piperazine Bioisosteres in the Olaparib Framework Shows Reduced DNA Damage and Cytotoxicity.

Reilly SW, Puentes LN, Wilson K, Hsieh CJ, Weng CC, Makvandi M, Mach RH. Reilly SW, et al. J Med Chem. 2018 Jun 28;61(12):5367-5379. doi: 10.1021/acs.jmedchem.8b00576. Epub 2018 Jun 14. J Med Chem. 2018. PMID: 29856625 Free PMC article.

8

Evaluation of a Low-Toxicity PARP Inhibitor as a Neuroprotective Agent for Parkinson's Disease.

Puentes LN, Lengyel-Zhand Z, Reilly SW, Mach RH. Puentes LN, et al. Among authors: reilly sw. Mol Neurobiol. 2021 Aug;58(8):3641-3652. doi: 10.1007/s12035-021-02371-4. Epub 2021 Mar 31. Mol Neurobiol. 2021. PMID: 33788167

9

Pd-Catalyzed Synthesis of Piperazine Scaffolds Under Aerobic and Solvent-Free Conditions.

Reilly SW, Mach RH. Reilly SW, et al. Org Lett. 2016 Oct 21;18(20):5272-5275. doi: 10.1021/acs.orglett.6b02591. Epub 2016 Oct 13. Org Lett. 2016. PMID: 27736075 Free PMC article.

10

Rapid Cu-Catalyzed [²¹¹At]Astatination and [¹²⁵I]Iodination of Boronic Esters at Room Temperature.

Reilly SW, Makvandi M, Xu K, Mach RH. Reilly SW, et al. Org Lett. 2018 Apr 6;20(7):1752-1755. doi: 10.1021/acs.orglett.8b00232. Epub 2018 Mar 21. Org Lett. 2018. PMID: 29561158 Free PMC article.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

17 results

Search Page