Frølund B - Search Results

1

Structure-Function Evaluation of Imidazopyridine Derivatives Selective for δ-Subunit-Containing γ-Aminobutyric Acid Type A (GABA_A) Receptors.

Yakoub K, Jung S, Sattler C, Damerow H, Weber J, Kretzschmann A, Cankaya AS, Piel M, Rösch F, Haugaard AS, Frølund B, Schirmeister T, Lüddens H. Yakoub K, et al. Among authors: frolund b. J Med Chem. 2018 Mar 8;61(5):1951-1968. doi: 10.1021/acs.jmedchem.7b01484. Epub 2018 Feb 26. J Med Chem. 2018. PMID: 29451785

2

Partial GABAA receptor agonists. Synthesis and in vitro pharmacology of a series of nonannulated analogs of 4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridin-3-ol.

Frølund B, Kristiansen U, Brehm L, Hansen AB, Krogsgaard-Larsen P, Falch E. Frølund B, et al. J Med Chem. 1995 Aug 18;38(17):3287-96. doi: 10.1021/jm00017a014. J Med Chem. 1995. PMID: 7650683

3

GABAA receptor agonists, partial agonists, and antagonists. Design and therapeutic prospects.

Krogsgaard-Larsen P, Frølund B, Jørgensen FS, Schousboe A. Krogsgaard-Larsen P, et al. Among authors: frolund b. J Med Chem. 1994 Aug 5;37(16):2489-505. doi: 10.1021/jm00042a001. J Med Chem. 1994. PMID: 8057295 Review. No abstract available.

4

A novel class of potent 3-isoxazolol GABA(A) antagonists: design, synthesis, and pharmacology.

Frølund B, Tagmose L, Liljefors T, Stensbøl TB, Engblom C, Kristiansen U, Krogsgaard-Larsen P. Frølund B, et al. J Med Chem. 2000 Dec 28;43(26):4930-3. doi: 10.1021/jm000371q. J Med Chem. 2000. PMID: 11150163 No abstract available.

5

Novel class of potent 4-arylalkyl substituted 3-isoxazolol GABA(A) antagonists: synthesis, pharmacology, and molecular modeling.

Frølund B, Jørgensen AT, Tagmose L, Stensbøl TB, Vestergaard HT, Engblom C, Kristiansen U, Sanchez C, Krogsgaard-Larsen P, Liljefors T. Frølund B, et al. J Med Chem. 2002 Jun 6;45(12):2454-68. doi: 10.1021/jm020027o. J Med Chem. 2002. PMID: 12036354

6

GABA(A) receptor ligands and their therapeutic potentials.

Frølund B, Ebert B, Kristiansen U, Liljefors T, Krogsgaard-Larsen P. Frølund B, et al. Curr Top Med Chem. 2002 Aug;2(8):817-32. doi: 10.2174/1568026023393525. Curr Top Med Chem. 2002. PMID: 12171573 Review.

7

Design and synthesis of a new series of 4-alkylated 3-isoxazolol GABA A antagonists.

Frølund B, Tagmose L, Jørgensen AT, Kristiansen U, Stensbøl TB, Liljefors T, Krogsgaard-Larsen P. Frølund B, et al. Eur J Med Chem. 2003 Apr;38(4):447-9. doi: 10.1016/s0223-5234(03)00056-4. Eur J Med Chem. 2003. PMID: 12750034

8

Aza-THIP and related analogues of THIP as GABA C antagonists.

Krehan D, Frølund B, Ebert B, Nielsen B, Krogsgaard-Larsen P, Johnston GA, Chebib M. Krehan D, et al. Among authors: frolund b. Bioorg Med Chem. 2003 Nov 17;11(23):4891-6. doi: 10.1016/j.bmc.2003.09.016. Bioorg Med Chem. 2003. PMID: 14604650

9

Selective inhibitors of GABA uptake: synthesis and molecular pharmacology of 4-N-methylamino-4,5,6,7-tetrahydrobenzo[d]isoxazol-3-ol analogues.

Clausen RP, Moltzen EK, Perregaard J, Lenz SM, Sanchez C, Falch E, Frølund B, Bolvig T, Sarup A, Larsson OM, Schousboe A, Krogsgaard-Larsen P. Clausen RP, et al. Among authors: frolund b. Bioorg Med Chem. 2005 Feb 1;13(3):895-908. doi: 10.1016/j.bmc.2004.10.029. Bioorg Med Chem. 2005. PMID: 15653355

10

Potent 4-aryl- or 4-arylalkyl-substituted 3-isoxazolol GABA(A) antagonists: synthesis, pharmacology, and molecular modeling.

Frølund B, Jensen LS, Guandalini L, Canillo C, Vestergaard HT, Kristiansen U, Nielsen B, Stensbøl TB, Madsen C, Krogsgaard-Larsen P, Liljefors T. Frølund B, et al. J Med Chem. 2005 Jan 27;48(2):427-39. doi: 10.1021/jm049256w. J Med Chem. 2005. PMID: 15658856

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