GABAA receptor agonists, partial agonists, and antagonists. Design and therapeutic prospects

J Med Chem. 1994 Aug 5;37(16):2489-505. doi: 10.1021/jm00042a001.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Animals
  • Drug Design
  • GABA Antagonists
  • Humans
  • Models, Molecular
  • Molecular Structure
  • Receptors, GABA / chemistry
  • Receptors, GABA / drug effects*
  • Receptors, GABA / physiology*
  • Recombinant Proteins / chemistry
  • Recombinant Proteins / metabolism
  • Structure-Activity Relationship
  • Therapeutics*
  • gamma-Aminobutyric Acid / chemistry
  • gamma-Aminobutyric Acid / physiology*

Substances

  • GABA Antagonists
  • Receptors, GABA
  • Recombinant Proteins
  • gamma-Aminobutyric Acid