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The Prodrug Approach: A Successful Tool for Improving Drug Solubility.
Molecules. 2015 Dec 29;21(1):42. doi: 10.3390/molecules21010042.
Molecules. 2015.
PMID: 26729077
Free PMC article.
Review.
Current Advances in Antitubercular Drug Discovery: Potent Prototypes and New Targets.
Dos Santos Fernandes GF, Jornada DH, de Souza PC, Chin CM, Pavan FR, Dos Santos JL.
Dos Santos Fernandes GF, et al.
Curr Med Chem. 2015;22(27):3133-61. doi: 10.2174/0929867322666150818103836.
Curr Med Chem. 2015.
PMID: 26282941
Review.
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Heterocyclic N-oxides - A Promising Class of Agents against Tuberculosis, Malaria and Neglected Tropical Diseases.
Dos Santos Fernandes GF, Pavan AR, Dos Santos JL.
Dos Santos Fernandes GF, et al.
Curr Pharm Des. 2018;24(12):1325-1340. doi: 10.2174/1381612824666180417122625.
Curr Pharm Des. 2018.
PMID: 29663875
Review.
Item in Clipboard
Design, Synthesis, and Characterization of N-Oxide-Containing Heterocycles with in Vivo Sterilizing Antitubercular Activity.
Dos Santos Fernandes GF, de Souza PC, Moreno-Viguri E, Santivañez-Veliz M, Paucar R, Pérez-Silanes S, Chegaev K, Guglielmo S, Lazzarato L, Fruttero R, Man Chin C, da Silva PB, Chorilli M, Solcia MC, Ribeiro CM, Silva CSP, Marino LB, Bosquesi PL, Hunt DM, de Carvalho LPS, de Souza Costa CA, Cho SH, Wang Y, Franzblau SG, Pavan FR, Dos Santos JL.
Dos Santos Fernandes GF, et al.
J Med Chem. 2017 Oct 26;60(20):8647-8660. doi: 10.1021/acs.jmedchem.7b01332. Epub 2017 Oct 16.
J Med Chem. 2017.
PMID: 28968083
Free PMC article.
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Tapping into the antitubercular potential of 2,5-dimethylpyrroles: A structure-activity relationship interrogation.
Semenya D, Touitou M, Masci D, Ribeiro CM, Pavan FR, Dos Santos Fernandes GF, Gianibbi B, Manetti F, Castagnolo D.
Semenya D, et al. Among authors: dos santos fernandes gf.
Eur J Med Chem. 2022 Jul 5;237:114404. doi: 10.1016/j.ejmech.2022.114404. Epub 2022 Apr 21.
Eur J Med Chem. 2022.
PMID: 35486992
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