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Antileishmanial Activity of 4,8-Dimethoxynaphthalenyl Chalcones on Leishmania amazonensis.
de Santiago-Silva KM, Bortoleti BTDS, Oliveira LDN, Maia FLA, Castro JC, Costa IC, Lazarin DB, Wardell JL, Wardell SMSV, Albuquerque MG, Lima CHDS, Pavanelli WR, Bispo MLF, Gonçalves RSB. de Santiago-Silva KM, et al. Antibiotics (Basel). 2022 Oct 13;11(10):1402. doi: 10.3390/antibiotics11101402. Antibiotics (Basel). 2022. PMID: 36290060 Free PMC article.
In silico approaches and in vitro assays identify a coumarin derivative as antiviral potential against SARS-CoV-2.
Felix da Silva Gomes G, Goes Camargo P, de Santiago-Silva KM, Suzukawa HT, Sotero da Silva Ribeiro AP, Orsato A, Nakazato G, Yamada-Ogatta SF, Faccin-Galhardi LC, da Silva Lima CH, de Lima Ferreira Bispo M, Perez CC. Felix da Silva Gomes G, et al. Among authors: de santiago silva km. J Biomol Struct Dyn. 2023 Oct-Nov;41(18):8978-8991. doi: 10.1080/07391102.2022.2140203. Epub 2022 Nov 3. J Biomol Struct Dyn. 2023. PMID: 36326347
Proteasome as a Drug Target in Trypanosomatid Diseases.
Silva ML, de Santiago-Silva KM, Fabris M, Camargo PG, de Lima Ferreira Bispo M. Silva ML, et al. Among authors: de santiago silva km. Curr Drug Targets. 2023;24(10):781-789. doi: 10.2174/1389450124666230719104147. Curr Drug Targets. 2023. PMID: 37469152
Molecular Targets for Chalcones in Antileishmanial Drug Discovery.
de Santiago-Silva KM, da Silva Gomes GF, Perez CC, da Silva Lima CH, de Lima Ferreira Bispo M. de Santiago-Silva KM, et al. Mini Rev Med Chem. 2023;23(14):1414-1434. doi: 10.2174/1389557523666230127125058. Mini Rev Med Chem. 2023. PMID: 36705240 Review.
CYP1B1: A Promising Target in Cancer Drug Discovery.
Fabris M, Luiza Silva M, de Santiago-Silva KM, de Lima Ferreira Bispo M, Goes Camargo P. Fabris M, et al. Among authors: de santiago silva km. Anticancer Agents Med Chem. 2023;23(9):981-988. doi: 10.2174/1871520623666230119103914. Anticancer Agents Med Chem. 2023. PMID: 36655529