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DNA binding and Topoisomerase inhibition: How can these mechanisms be explored to design more specific anticancer agents?
de Almeida SMV, Ribeiro AG, de Lima Silva GC, Ferreira Alves JE, Beltrão EIC, de Oliveira JF, de Carvalho LB Junior, Alves de Lima MDC. de Almeida SMV, et al. Among authors: de carvalho lb junior, de lima silva gc, de oliveira jf. Biomed Pharmacother. 2017 Dec;96:1538-1556. doi: 10.1016/j.biopha.2017.11.054. Epub 2017 Nov 22. Biomed Pharmacother. 2017. PMID: 29174576 Review.
In vivo study of schistosomicidal action of 1-benzyl-4-[(4-fluoro-phenyl)-hydrazono]-5-thioxo-imidazolidin-2-one.
da Silva AL, de Oliveira JF, Silva WL, Luis AF, de Farias Santiago E, Alves de Almeida Júnior AS, de Oliveira TB, de Souza VCA, de Barros AF, Pitta IDR, de Oliveira SA, Alves de Lima MDC. da Silva AL, et al. Among authors: de barros af, de souza vca, de farias santiago e, de oliveira tb, de oliveira sa, de oliveira jf. Biomed Pharmacother. 2016 Oct;83:502-507. doi: 10.1016/j.biopha.2016.07.008. Epub 2016 Jul 18. Biomed Pharmacother. 2016. PMID: 27434866
Thiosemicarbazones and 4-thiazolidinones indole-based derivatives: Synthesis, evaluation of antiproliferative activity, cell death mechanisms and topoisomerase inhibition assay.
de Oliveira JF, Lima TS, Vendramini-Costa DB, de Lacerda Pedrosa SCB, Lafayette EA, da Silva RMF, de Almeida SMV, de Moura RO, Ruiz ALTG, de Carvalho JE, de Lima MDCA. de Oliveira JF, et al. Among authors: de almeida smv, de moura ro, de lacerda pedrosa scb, de carvalho je, de lima mdca. Eur J Med Chem. 2017 Aug 18;136:305-314. doi: 10.1016/j.ejmech.2017.05.023. Epub 2017 May 8. Eur J Med Chem. 2017. PMID: 28505535
Synthesis of novel indole derivatives as promising DNA-binding agents and evaluation of antitumor and antitopoisomerase I activities.
Lafayette EA, de Almeida SMV, Cavalcanti Santos RV, de Oliveira JF, Amorim CADC, da Silva RMF, Pitta MGDR, Pitta IDR, de Moura RO, de Carvalho Júnior LB, de Melo Rêgo MJB, de Lima MDCA. Lafayette EA, et al. Among authors: de almeida smv, de moura ro, de carvalho junior lb, de melo rego mjb, de oliveira jf, de lima mdca. Eur J Med Chem. 2017 Aug 18;136:511-522. doi: 10.1016/j.ejmech.2017.05.012. Epub 2017 May 4. Eur J Med Chem. 2017. PMID: 28531811
New thiophene-acridine compounds: Synthesis, antileishmanial activity, DNA binding, chemometric, and molecular docking studies.
de Lima Serafim V, Félix MB, Frade Silva DK, Rodrigues KADF, Andrade PN, de Almeida SMV, de Albuquerque Dos Santos S, de Oliveira JF, de Lima MDCA, Mendonça-Junior FJB, Scotti MT, de Oliveira MR, de Moura RO. de Lima Serafim V, et al. Among authors: de almeida smv, de moura ro, de albuquerque dos santos s, de oliveira mr, de oliveira jf, de lima mdca. Chem Biol Drug Des. 2018 Jun;91(6):1141-1155. doi: 10.1111/cbdd.13176. Epub 2018 Mar 25. Chem Biol Drug Des. 2018. PMID: 29415325
Synthesis, DNA and protein interactions and human topoisomerase inhibition of novel Spiroacridine derivatives.
Gouveia RG, Ribeiro AG, Segundo MÂSP, de Oliveira JF, de Lima MDCA, de Lima Souza TRC, de Almeida SMV, de Moura RO. Gouveia RG, et al. Among authors: de almeida smv, de moura ro, de lima souza trc, de oliveira jf, de lima mdca. Bioorg Med Chem. 2018 Dec 1;26(22):5911-5921. doi: 10.1016/j.bmc.2018.10.038. Epub 2018 Oct 29. Bioorg Med Chem. 2018. PMID: 30420325
Topoisomerase inhibition and albumin interaction studies of acridine-thiosemicarbazone derivatives.
da Silva Filho FA, de Freitas Souza T, Ribeiro AG, Alves JEF, de Oliveira JF, de Lima Souza TRC, de Moura RO, do Carmo Alves de Lima M, de Carvalho Junior LB, de Almeida SMV. da Silva Filho FA, et al. Among authors: de almeida smv, de moura ro, de carvalho junior lb, de freitas souza t, de lima souza trc, de oliveira jf. Int J Biol Macromol. 2019 Oct 1;138:582-589. doi: 10.1016/j.ijbiomac.2019.07.097. Epub 2019 Jul 16. Int J Biol Macromol. 2019. PMID: 31323270 Free article.
Novel 4-quinoline-thiosemicarbazone derivatives: Synthesis, antiproliferative activity, in vitro and in silico biomacromolecule interaction studies and topoisomerase inhibition.
Ribeiro AG, Almeida SMV, de Oliveira JF, Souza TRCL, Santos KLD, Albuquerque APB, Nogueira MCBL, Carvalho Junior LB, Moura RO, da Silva AC, Pereira VRA, Castro MCAB, Lima MDCA. Ribeiro AG, et al. Among authors: de oliveira jf. Eur J Med Chem. 2019 Nov 15;182:111592. doi: 10.1016/j.ejmech.2019.111592. Epub 2019 Aug 6. Eur J Med Chem. 2019. PMID: 31421632
138 results