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ACW-02 an Acridine Triazolidine Derivative Presents Antileishmanial Activity Mediated by DNA Interaction and Immunomodulation.
Albino SL, da Silva Moura WC, Reis MMLD, Sousa GLS, da Silva PR, de Oliveira MGC, Borges TKDS, Albuquerque LFF, de Almeida SMV, de Lima MDCA, Kuckelhaus SAS, Nascimento IJDS, Junior FJBM, da Silva TG, de Moura RO. Albino SL, et al. Among authors: de moura ro. Pharmaceuticals (Basel). 2023 Jan 29;16(2):204. doi: 10.3390/ph16020204. Pharmaceuticals (Basel). 2023. PMID: 37259353 Free PMC article.
Synthesis, DNA Binding, and Antiproliferative Activity of Novel Acridine-Thiosemicarbazone Derivatives.
de Almeida SM, Lafayette EA, da Silva LP, Amorim CA, de Oliveira TB, Ruiz AL, de Carvalho JE, de Moura RO, Beltrão EI, de Lima Mdo C, de Carvalho Júnior LB. de Almeida SM, et al. Among authors: de moura ro, de carvalho junior lb, de lima mdo c, de oliveira tb, de carvalho je. Int J Mol Sci. 2015 Jun 9;16(6):13023-42. doi: 10.3390/ijms160613023. Int J Mol Sci. 2015. PMID: 26068233 Free PMC article.
2-Amino-thiophene derivatives present antileishmanial activity mediated by apoptosis and immunomodulation in vitro.
Rodrigues KA, Dias CN, Néris PL, Rocha Jda C, Scotti MT, Scotti L, Mascarenhas SR, Veras RC, de Medeiros IA, Keesen Tde S, de Oliveira TB, de Lima Mdo C, Balliano TL, de Aquino TM, de Moura RO, Mendonça Junior FJ, de Oliveira MR. Rodrigues KA, et al. Among authors: de moura ro, de aquino tm, de lima mdo c, de oliveira mr, de oliveira tb, de medeiros ia. Eur J Med Chem. 2015 Dec 1;106:1-14. doi: 10.1016/j.ejmech.2015.10.011. Epub 2015 Oct 17. Eur J Med Chem. 2015. PMID: 26513640
Thiosemicarbazones and 4-thiazolidinones indole-based derivatives: Synthesis, evaluation of antiproliferative activity, cell death mechanisms and topoisomerase inhibition assay.
de Oliveira JF, Lima TS, Vendramini-Costa DB, de Lacerda Pedrosa SCB, Lafayette EA, da Silva RMF, de Almeida SMV, de Moura RO, Ruiz ALTG, de Carvalho JE, de Lima MDCA. de Oliveira JF, et al. Among authors: de almeida smv, de moura ro, de lacerda pedrosa scb, de carvalho je, de lima mdca. Eur J Med Chem. 2017 Aug 18;136:305-314. doi: 10.1016/j.ejmech.2017.05.023. Epub 2017 May 8. Eur J Med Chem. 2017. PMID: 28505535
Synthesis of novel indole derivatives as promising DNA-binding agents and evaluation of antitumor and antitopoisomerase I activities.
Lafayette EA, de Almeida SMV, Cavalcanti Santos RV, de Oliveira JF, Amorim CADC, da Silva RMF, Pitta MGDR, Pitta IDR, de Moura RO, de Carvalho Júnior LB, de Melo Rêgo MJB, de Lima MDCA. Lafayette EA, et al. Among authors: de almeida smv, de moura ro, de carvalho junior lb, de melo rego mjb, de oliveira jf, de lima mdca. Eur J Med Chem. 2017 Aug 18;136:511-522. doi: 10.1016/j.ejmech.2017.05.012. Epub 2017 May 4. Eur J Med Chem. 2017. PMID: 28531811
New thiophene-acridine compounds: Synthesis, antileishmanial activity, DNA binding, chemometric, and molecular docking studies.
de Lima Serafim V, Félix MB, Frade Silva DK, Rodrigues KADF, Andrade PN, de Almeida SMV, de Albuquerque Dos Santos S, de Oliveira JF, de Lima MDCA, Mendonça-Junior FJB, Scotti MT, de Oliveira MR, de Moura RO. de Lima Serafim V, et al. Among authors: de almeida smv, de moura ro, de albuquerque dos santos s, de oliveira mr, de oliveira jf, de lima mdca. Chem Biol Drug Des. 2018 Jun;91(6):1141-1155. doi: 10.1111/cbdd.13176. Epub 2018 Mar 25. Chem Biol Drug Des. 2018. PMID: 29415325
Synthesis, DNA and protein interactions and human topoisomerase inhibition of novel Spiroacridine derivatives.
Gouveia RG, Ribeiro AG, Segundo MÂSP, de Oliveira JF, de Lima MDCA, de Lima Souza TRC, de Almeida SMV, de Moura RO. Gouveia RG, et al. Among authors: de almeida smv, de moura ro, de lima souza trc, de oliveira jf, de lima mdca. Bioorg Med Chem. 2018 Dec 1;26(22):5911-5921. doi: 10.1016/j.bmc.2018.10.038. Epub 2018 Oct 29. Bioorg Med Chem. 2018. PMID: 30420325
Topoisomerase inhibition and albumin interaction studies of acridine-thiosemicarbazone derivatives.
da Silva Filho FA, de Freitas Souza T, Ribeiro AG, Alves JEF, de Oliveira JF, de Lima Souza TRC, de Moura RO, do Carmo Alves de Lima M, de Carvalho Junior LB, de Almeida SMV. da Silva Filho FA, et al. Among authors: de almeida smv, de moura ro, de carvalho junior lb, de freitas souza t, de lima souza trc, de oliveira jf. Int J Biol Macromol. 2019 Oct 1;138:582-589. doi: 10.1016/j.ijbiomac.2019.07.097. Epub 2019 Jul 16. Int J Biol Macromol. 2019. PMID: 31323270 Free article.
Bioprospecting of Nitrogenous Heterocyclic Scaffolds with Potential Action for Neglected Parasitosis: A Review.
Albino SL, da Silva JM, de C Nobre MS, de M E Silva YMS, Santos MB, de Araújo RSA, do C A de Lima M, Schmitt M, de Moura RO. Albino SL, et al. Among authors: de moura ro, de araujo rsa, de c nobre ms, de m e silva yms. Curr Pharm Des. 2020;26(33):4112-4150. doi: 10.2174/1381612826666200701160904. Curr Pharm Des. 2020. PMID: 32611290 Free article. Review.
44 results