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New thiophene-acridine compounds: Synthesis, antileishmanial activity, DNA binding, chemometric, and molecular docking studies.
de Lima Serafim V, Félix MB, Frade Silva DK, Rodrigues KADF, Andrade PN, de Almeida SMV, de Albuquerque Dos Santos S, de Oliveira JF, de Lima MDCA, Mendonça-Junior FJB, Scotti MT, de Oliveira MR, de Moura RO. de Lima Serafim V, et al. Among authors: de almeida smv, de moura ro, de albuquerque dos santos s, de oliveira mr, de oliveira jf, de lima mdca. Chem Biol Drug Des. 2018 Jun;91(6):1141-1155. doi: 10.1111/cbdd.13176. Epub 2018 Mar 25. Chem Biol Drug Des. 2018. PMID: 29415325
Synthesis, structure-activity relationships (SAR) and in silico studies of coumarin derivatives with antifungal activity.
de Araújo RS, Guerra FQ, de O Lima E, de Simone CA, Tavares JF, Scotti L, Scotti MT, de Aquino TM, de Moura RO, Mendonça FJ, Barbosa-Filho JM. de Araújo RS, et al. Among authors: de moura ro, de aquino tm, de simone ca, de o lima e. Int J Mol Sci. 2013 Jan 10;14(1):1293-309. doi: 10.3390/ijms14011293. Int J Mol Sci. 2013. PMID: 23306152 Free PMC article.
Synthesis, DNA Binding, and Antiproliferative Activity of Novel Acridine-Thiosemicarbazone Derivatives.
de Almeida SM, Lafayette EA, da Silva LP, Amorim CA, de Oliveira TB, Ruiz AL, de Carvalho JE, de Moura RO, Beltrão EI, de Lima Mdo C, de Carvalho Júnior LB. de Almeida SM, et al. Among authors: de moura ro, de carvalho junior lb, de lima mdo c, de oliveira tb, de carvalho je. Int J Mol Sci. 2015 Jun 9;16(6):13023-42. doi: 10.3390/ijms160613023. Int J Mol Sci. 2015. PMID: 26068233 Free PMC article.
2-Amino-thiophene derivatives present antileishmanial activity mediated by apoptosis and immunomodulation in vitro.
Rodrigues KA, Dias CN, Néris PL, Rocha Jda C, Scotti MT, Scotti L, Mascarenhas SR, Veras RC, de Medeiros IA, Keesen Tde S, de Oliveira TB, de Lima Mdo C, Balliano TL, de Aquino TM, de Moura RO, Mendonça Junior FJ, de Oliveira MR. Rodrigues KA, et al. Among authors: de moura ro, de aquino tm, de lima mdo c, de oliveira mr, de oliveira tb, de medeiros ia. Eur J Med Chem. 2015 Dec 1;106:1-14. doi: 10.1016/j.ejmech.2015.10.011. Epub 2015 Oct 17. Eur J Med Chem. 2015. PMID: 26513640
Multi-Target Drugs for Neglected Diseases.
Scotti L, Filho FJ, de Moura RO, Ribeiro FF, Ishiki H, da Silva MS, Filho JM, Scotti MT. Scotti L, et al. Among authors: de moura ro. Curr Pharm Des. 2016 May 30;22(21):3135-63. doi: 10.2174/1381612822666160224142552. Curr Pharm Des. 2016. PMID: 26907943 Review.
Hybrid Compounds as Direct Multitarget Ligands: A Review.
de Oliveira Pedrosa M, Duarte da Cruz RM, de Oliveira Viana J, de Moura RO, Ishiki HM, Barbosa Filho JM, Diniz MF, Scotti MT, Scotti L, Bezerra Mendonca FJ. de Oliveira Pedrosa M, et al. Among authors: de oliveira viana j, de moura ro. Curr Top Med Chem. 2017;17(9):1044-1079. doi: 10.2174/1568026616666160927160620. Curr Top Med Chem. 2017. PMID: 27697048 Review.
Thiosemicarbazones and 4-thiazolidinones indole-based derivatives: Synthesis, evaluation of antiproliferative activity, cell death mechanisms and topoisomerase inhibition assay.
de Oliveira JF, Lima TS, Vendramini-Costa DB, de Lacerda Pedrosa SCB, Lafayette EA, da Silva RMF, de Almeida SMV, de Moura RO, Ruiz ALTG, de Carvalho JE, de Lima MDCA. de Oliveira JF, et al. Among authors: de almeida smv, de moura ro, de lacerda pedrosa scb, de carvalho je, de lima mdca. Eur J Med Chem. 2017 Aug 18;136:305-314. doi: 10.1016/j.ejmech.2017.05.023. Epub 2017 May 8. Eur J Med Chem. 2017. PMID: 28505535
Synthesis of novel indole derivatives as promising DNA-binding agents and evaluation of antitumor and antitopoisomerase I activities.
Lafayette EA, de Almeida SMV, Cavalcanti Santos RV, de Oliveira JF, Amorim CADC, da Silva RMF, Pitta MGDR, Pitta IDR, de Moura RO, de Carvalho Júnior LB, de Melo Rêgo MJB, de Lima MDCA. Lafayette EA, et al. Among authors: de almeida smv, de moura ro, de carvalho junior lb, de melo rego mjb, de oliveira jf, de lima mdca. Eur J Med Chem. 2017 Aug 18;136:511-522. doi: 10.1016/j.ejmech.2017.05.012. Epub 2017 May 4. Eur J Med Chem. 2017. PMID: 28531811
44 results