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Discovery of MK-8970: an acetal carbonate prodrug of raltegravir with enhanced colonic absorption.
ChemMedChem. 2015 Feb;10(2):245-52. doi: 10.1002/cmdc.201402393. Epub 2014 Dec 2.
ChemMedChem. 2015.
PMID: 25469982
Synthesis of a CGRP Receptor Antagonist via an Asymmetric Synthesis of 3-Fluoro-4-aminopiperidine.
Molinaro C, Phillips EM, Xiang B, Milczek E, Shevlin M, Balsells J, Ceglia S, Chen J, Chen L, Chen Q, Fei Z, Hoerrner S, Qi J, de Lera Ruiz M, Tan L, Wan B, Yin J.
Molinaro C, et al. Among authors: de lera ruiz m.
J Org Chem. 2019 Jun 21;84(12):8006-8018. doi: 10.1021/acs.joc.9b00569. Epub 2019 Jun 5.
J Org Chem. 2019.
PMID: 31124362
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Bicyclic and tricyclic heterocycle derivatives as histamine H3 receptor antagonists for the treatment of obesity.
de Lera Ruiz M, Zheng J, Berlin MY, McCormick KD, Aslanian RG, West R, Hwa J, Lachowicz J, van Heek M.
de Lera Ruiz M, et al.
Bioorg Med Chem Lett. 2013 Nov 1;23(21):6004-9. doi: 10.1016/j.bmcl.2013.08.013. Epub 2013 Aug 19.
Bioorg Med Chem Lett. 2013.
PMID: 24035485
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Adenosine A2A receptor as a drug discovery target.
de Lera Ruiz M, Lim YH, Zheng J.
de Lera Ruiz M, et al.
J Med Chem. 2014 May 8;57(9):3623-50. doi: 10.1021/jm4011669. Epub 2013 Nov 15.
J Med Chem. 2014.
PMID: 24164628
Review.
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Voltage-Gated Sodium Channels: Structure, Function, Pharmacology, and Clinical Indications.
de Lera Ruiz M, Kraus RL.
de Lera Ruiz M, et al.
J Med Chem. 2015 Sep 24;58(18):7093-118. doi: 10.1021/jm501981g. Epub 2015 May 14.
J Med Chem. 2015.
PMID: 25927480
Review.
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The Invention of WM382, a Highly Potent PMIX/X Dual Inhibitor toward the Treatment of Malaria.
de Lera Ruiz M, Favuzza P, Guo Z, Zhao L, Hu B, Lei Z, Zhan D, Murgolo N, Boyce CW, Vavrek M, Thompson J, Ngo A, Jarman KE, Robbins J, Boddey J, Sleebs BE, Lowes KN, Cowman AF, Olsen DB, McCauley JA.
de Lera Ruiz M, et al.
ACS Med Chem Lett. 2022 Oct 12;13(11):1745-1754. doi: 10.1021/acsmedchemlett.2c00355. eCollection 2022 Nov 10.
ACS Med Chem Lett. 2022.
PMID: 36385924
Free PMC article.
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Dual Plasmepsin-Targeting Antimalarial Agents Disrupt Multiple Stages of the Malaria Parasite Life Cycle.
Favuzza P, de Lera Ruiz M, Thompson JK, Triglia T, Ngo A, Steel RWJ, Vavrek M, Christensen J, Healer J, Boyce C, Guo Z, Hu M, Khan T, Murgolo N, Zhao L, Penington JS, Reaksudsan K, Jarman K, Dietrich MH, Richardson L, Guo KY, Lopaticki S, Tham WH, Rottmann M, Papenfuss T, Robbins JA, Boddey JA, Sleebs BE, Sabroux HJ, McCauley JA, Olsen DB, Cowman AF.
Favuzza P, et al. Among authors: de lera ruiz m.
Cell Host Microbe. 2020 Apr 8;27(4):642-658.e12. doi: 10.1016/j.chom.2020.02.005. Epub 2020 Feb 27.
Cell Host Microbe. 2020.
PMID: 32109369
Free PMC article.
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Invention of MK-7845, a SARS-CoV-2 3CL Protease Inhibitor Employing a Novel Difluorinated Glutamine Mimic.
Shurtleff VW, Layton ME, Parish CA, Perkins JJ, Schreier JD, Wang Y, Adam GC, Alvarez N, Bahmanjah S, Bahnck-Teets CM, Boyce CW, Burlein C, Cabalu TD, Campbell BT, Carroll SS, Chang W, de Lera Ruiz M, Dolgov E, Fay JF, Fox NG, Goh SL, Hartingh TJ, Hurzy DM, Kelly MJ 3rd, Klein DJ, Klingler FM, Krishnamurthy H, Kudalkar S, Mayhood TW, McKenna PM, Murray EM, Nahas D, Nawrat CC, Park S, Qian D, Roecker AJ, Sharma V, Shipe WD, Su J, Taggart RV, Truong Q, Wu Y, Zhou X, Zhuang N, Perlin DS, Olsen DB, Howe JA, McCauley JA.
Shurtleff VW, et al. Among authors: de lera ruiz m.
J Med Chem. 2024 Mar 14;67(5):3935-3958. doi: 10.1021/acs.jmedchem.3c02248. Epub 2024 Feb 16.
J Med Chem. 2024.
PMID: 38365209
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