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A multitarget approach to drug discovery inhibiting Mycobacterium tuberculosis PyrG and PanK.
Sci Rep. 2018 Feb 16;8(1):3187. doi: 10.1038/s41598-018-21614-4.
Sci Rep. 2018.
PMID: 29453370
Free PMC article.
Thiophenecarboxamide Derivatives Activated by EthA Kill Mycobacterium tuberculosis by Inhibiting the CTP Synthetase PyrG.
Mori G, Chiarelli LR, Esposito M, Makarov V, Bellinzoni M, Hartkoorn RC, Degiacomi G, Boldrin F, Ekins S, de Jesus Lopes Ribeiro AL, Marino LB, Centárová I, Svetlíková Z, Blaško J, Kazakova E, Lepioshkin A, Barilone N, Zanoni G, Porta A, Fondi M, Fani R, Baulard AR, Mikušová K, Alzari PM, Manganelli R, de Carvalho LP, Riccardi G, Cole ST, Pasca MR.
Mori G, et al. Among authors: de jesus lopes ribeiro al.
Chem Biol. 2015 Jul 23;22(7):917-27. doi: 10.1016/j.chembiol.2015.05.016. Epub 2015 Jun 18.
Chem Biol. 2015.
PMID: 26097035
Free PMC article.
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Antituberculars which target decaprenylphosphoryl-β-D-ribofuranose 2'-oxidase DprE1: state of art.
Buroni S, Pasca MR, de Jesus Lopes Ribeiro AL, Degiacomi G, Molteni E, Riccardi G.
Buroni S, et al. Among authors: de jesus lopes ribeiro al.
Appl Microbiol Biotechnol. 2012 May;94(4):907-16. doi: 10.1007/s00253-012-4013-4. Epub 2012 Apr 18.
Appl Microbiol Biotechnol. 2012.
PMID: 22526781
Retracted.
Review.
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DprE1, a new taxonomic marker in mycobacteria.
Incandela ML, Perrin E, Fondi M, de Jesus Lopes Ribeiro AL, Mori G, Moiana A, Gramegna M, Fani R, Riccardi G, Pasca MR.
Incandela ML, et al. Among authors: de jesus lopes ribeiro al.
FEMS Microbiol Lett. 2013 Nov;348(1):66-73. doi: 10.1111/1574-6968.12246. Epub 2013 Sep 12.
FEMS Microbiol Lett. 2013.
PMID: 24024613
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2-Carboxyquinoxalines kill mycobacterium tuberculosis through noncovalent inhibition of DprE1.
Neres J, Hartkoorn RC, Chiarelli LR, Gadupudi R, Pasca MR, Mori G, Venturelli A, Savina S, Makarov V, Kolly GS, Molteni E, Binda C, Dhar N, Ferrari S, Brodin P, Delorme V, Landry V, de Jesus Lopes Ribeiro AL, Farina D, Saxena P, Pojer F, Carta A, Luciani R, Porta A, Zanoni G, De Rossi E, Costi MP, Riccardi G, Cole ST.
Neres J, et al. Among authors: de jesus lopes ribeiro al.
ACS Chem Biol. 2015 Mar 20;10(3):705-14. doi: 10.1021/cb5007163. Epub 2014 Dec 9.
ACS Chem Biol. 2015.
PMID: 25427196
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Evaluation of fluoroquinolone resistance mechanisms in Pseudomonas aeruginosa multidrug resistance clinical isolates.
Pasca MR, Dalla Valle C, De Jesus Lopes Ribeiro AL, Buroni S, Papaleo MC, Bazzini S, Udine C, Incandela ML, Daffara S, Fani R, Riccardi G, Marone P.
Pasca MR, et al. Among authors: de jesus lopes ribeiro al.
Microb Drug Resist. 2012 Feb;18(1):23-32. doi: 10.1089/mdr.2011.0019. Epub 2011 Jul 28.
Microb Drug Resist. 2012.
PMID: 21797666
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Design, chemical synthesis of 3-(9H-fluoren-9-yl)pyrrolidine-2,5-dione derivatives and biological activity against enoyl-ACP reductase (InhA) and Mycobacterium tuberculosis.
Matviiuk T, Rodriguez F, Saffon N, Mallet-Ladeira S, Gorichko M, de Jesus Lopes Ribeiro AL, Pasca MR, Lherbet C, Voitenko Z, Baltas M.
Matviiuk T, et al. Among authors: de jesus lopes ribeiro al.
Eur J Med Chem. 2013;70:37-48. doi: 10.1016/j.ejmech.2013.09.041. Epub 2013 Oct 2.
Eur J Med Chem. 2013.
PMID: 24140915
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