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Page 1
Current advances in drug discovery for Chagas disease.
Scarim CB, Jornada DH, Chelucci RC, de Almeida L, Dos Santos JL, Chung MC. Scarim CB, et al. Among authors: de almeida l. Eur J Med Chem. 2018 Jul 15;155:824-838. doi: 10.1016/j.ejmech.2018.06.040. Epub 2018 Jun 20. Eur J Med Chem. 2018. PMID: 30033393 Review.
In vivo antileishmanial activity and histopathological evaluation in Leishmania infantum infected hamsters after treatment with a furoxan derivative.
de Almeida L, Passalacqua TG, Dutra LA, Fonseca JNVD, Nascimento RFQ, Imamura KB, de Andrade CR, Dos Santos JL, Graminha MAS. de Almeida L, et al. Among authors: de andrade cr. Biomed Pharmacother. 2017 Nov;95:536-547. doi: 10.1016/j.biopha.2017.08.096. Epub 2017 Sep 12. Biomed Pharmacother. 2017. PMID: 28866421
Leishmanicidal activities of novel synthetic furoxan and benzofuroxan derivatives.
Dutra LA, de Almeida L, Passalacqua TG, Reis JS, Torres FA, Martinez I, Peccinini RG, Chin CM, Chegaev K, Guglielmo S, Fruttero R, Graminha MA, dos Santos JL. Dutra LA, et al. Among authors: de almeida l. Antimicrob Agents Chemother. 2014 Aug;58(8):4837-47. doi: 10.1128/AAC.00052-14. Epub 2014 Jun 9. Antimicrob Agents Chemother. 2014. PMID: 24913171 Free PMC article.
Synthesis and evaluation of novel prenylated chalcone derivatives as anti-leishmanial and anti-trypanosomal compounds.
Passalacqua TG, Dutra LA, de Almeida L, Velásquez AM, Torres FA, Yamasaki PR, dos Santos MB, Regasini LO, Michels PA, Bolzani Vda S, Graminha MA. Passalacqua TG, et al. Among authors: de almeida l. Bioorg Med Chem Lett. 2015 Aug 15;25(16):3342-5. doi: 10.1016/j.bmcl.2015.05.072. Epub 2015 May 30. Bioorg Med Chem Lett. 2015. PMID: 26055530
The 2',4'-dihydroxychalcone could be explored to develop new inhibitors against the glycerol-3-phosphate dehydrogenase from Leishmania species.
Passalacqua TG, Torres FA, Nogueira CT, de Almeida L, Del Cistia ML, dos Santos MB, Dutra LA, Bolzani VS, Regasini LO, Graminha MA, Marchetto R, Zottis A. Passalacqua TG, et al. Among authors: de almeida l. Bioorg Med Chem Lett. 2015 Sep 1;25(17):3564-8. doi: 10.1016/j.bmcl.2015.06.085. Epub 2015 Jun 30. Bioorg Med Chem Lett. 2015. PMID: 26169126
Corrigendum to "The 2',4'-dihydroxychalcone could be explored to develop new inhibitors against the glycerol-3-phosphate dehydrogenase from Leishmania species" [Bioorg. Med. Chem. Lett. 25 (2015) 3564-3568].
Passalacqua TG, Torres FAE, Nogueira CT, de Almeida L, Del Cistia ML, Dos Santos MB, Dutra LA, da Silva Bolzani V, Regasini LO, Graminha MAS, Marchetto R, Zottis A. Passalacqua TG, et al. Among authors: de almeida l. Bioorg Med Chem Lett. 2017 May 1;27(9):2080. doi: 10.1016/j.bmcl.2017.03.044. Epub 2017 Mar 28. Bioorg Med Chem Lett. 2017. PMID: 28363747 No abstract available.
Nanotechnological Strategies for Treatment of Leishmaniasis--A Review.
de Almeida L, Terumi Fujimura A, Del Cistia ML, Fonseca-Santos B, Braga Imamura K, Michels PAM, Chorilli M, Graminha MAS. de Almeida L, et al. J Biomed Nanotechnol. 2017 Feb;13(2):117-33. doi: 10.1166/jbn.2017.2349. J Biomed Nanotechnol. 2017. PMID: 29376626 Review.
621 results