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Integrating synthetic accessibility with AI-based generative drug design.
J Cheminform. 2023 Sep 19;15(1):83. doi: 10.1186/s13321-023-00742-8.
J Cheminform. 2023.
PMID: 37726842
Free PMC article.
Could we expect new praziquantel derivatives? A meta pharmacometrics/pharmacoinformatics analysis of all antischistosomal praziquantel derivatives found in the literature.
da Silva VBR, Boucherle B, El-Methni J, Hoffmann B, da Silva AL, Fortune A, de Lima MDCA, Thomas A.
da Silva VBR, et al.
SAR QSAR Environ Res. 2019 Jun;30(6):383-401. doi: 10.1080/1062936X.2019.1607898.
SAR QSAR Environ Res. 2019.
PMID: 31144535
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Medicinal chemistry of antischistosomal drugs: Praziquantel and oxamniquine.
da Silva VBR, Campos BRKL, de Oliveira JF, Decout JL, do Carmo Alves de Lima M.
da Silva VBR, et al.
Bioorg Med Chem. 2017 Jul 1;25(13):3259-3277. doi: 10.1016/j.bmc.2017.04.031. Epub 2017 Apr 27.
Bioorg Med Chem. 2017.
PMID: 28495384
Review.
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