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Comparative structural analyses of the NHL domains from the human E3 ligase TRIM-NHL family.
IUCrJ. 2022 Sep 27;9(Pt 6):720-727. doi: 10.1107/S2052252522008582. eCollection 2022 Nov 1.
IUCrJ. 2022.
PMID: 36381143
Free PMC article.
Propranolol Activates the Orphan Nuclear Receptor TLX to Counteract Proliferation and Migration of Glioblastoma Cells.
Faudone G, Bischoff-Kont I, Rachor L, Willems S, Zhubi R, Kaiser A, Chaikuad A, Knapp S, Fürst R, Heering J, Merk D.
Faudone G, et al. Among authors: zhubi r.
J Med Chem. 2021 Jun 24;64(12):8727-8738. doi: 10.1021/acs.jmedchem.1c00733. Epub 2021 Jun 11.
J Med Chem. 2021.
PMID: 34115934
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Design of a Potent TLX Agonist by Rational Fragment Fusion.
Faudone G, Zhubi R, Celik F, Knapp S, Chaikuad A, Heering J, Merk D.
Faudone G, et al. Among authors: zhubi r.
J Med Chem. 2022 Feb 10;65(3):2288-2296. doi: 10.1021/acs.jmedchem.1c01757. Epub 2022 Jan 6.
J Med Chem. 2022.
PMID: 34989568
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Kinase domain autophosphorylation rewires the activity and substrate specificity of CK1 enzymes.
Cullati SN, Chaikuad A, Chen JS, Gebel J, Tesmer L, Zhubi R, Navarrete-Perea J, Guillen RX, Gygi SP, Hummer G, Dötsch V, Knapp S, Gould KL.
Cullati SN, et al. Among authors: zhubi r.
Mol Cell. 2022 Jun 2;82(11):2006-2020.e8. doi: 10.1016/j.molcel.2022.03.005. Epub 2022 Mar 29.
Mol Cell. 2022.
PMID: 35353987
Free PMC article.
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Fragment-based discovery of orphan nuclear receptor Nur77/NGFI-B ligands.
Arifi S, Zaienne D, Heering J, Wein T, Zhubi R, Chaikuad A, Knapp S, Marschner JA, Merk D.
Arifi S, et al. Among authors: zhubi r.
Bioorg Chem. 2022 Dec;129:106164. doi: 10.1016/j.bioorg.2022.106164. Epub 2022 Sep 17.
Bioorg Chem. 2022.
PMID: 36162288
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Shifting the selectivity of pyrido[2,3-d]pyrimidin-7(8H)-one inhibitors towards the salt-inducible kinase (SIK) subfamily.
Rak M, Tesch R, Berger LM, Shevchenko E, Raab M, Tjaden A, Zhubi R, Balourdas DI, Joerger AC, Poso A, Krämer A, Elson L, Lučić A, Kronenberger T, Hanke T, Strebhardt K, Sanhaji M, Knapp S.
Rak M, et al. Among authors: zhubi r.
Eur J Med Chem. 2023 Jun 5;254:115347. doi: 10.1016/j.ejmech.2023.115347. Epub 2023 Apr 7.
Eur J Med Chem. 2023.
PMID: 37094449
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Back-pocket optimization of 2-aminopyrimidine-based macrocycles leads to potent dual EPHA2/GAK kinase inhibitors with antiviral activity.
Gerninghaus J, Zhubi R, Krämer A, Karim M, Tran DHN, Joerger AC, Schreiber C, Berger LM, Berger BT, Ehret TAL, Elson L, Lenz C, Saxena K, Müller S, Einav S, Knapp S, Hanke T.
Gerninghaus J, et al. Among authors: zhubi r.
bioRxiv [Preprint]. 2024 Feb 18:2024.02.18.580805. doi: 10.1101/2024.02.18.580805.
bioRxiv. 2024.
PMID: 38405908
Free PMC article.
Preprint.
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