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Drug Design Strategies to Avoid Resistance in Direct-Acting Antivirals and Beyond.
Chem Rev. 2021 Mar 24;121(6):3238-3270. doi: 10.1021/acs.chemrev.0c00648. Epub 2021 Jan 7.
Chem Rev. 2021.
PMID: 33410674
Free PMC article.
Review.
Hepatitis C Virus NS3/4A Protease Inhibitors Incorporating Flexible P2 Quinoxalines Target Drug Resistant Viral Variants.
Matthew AN, Zephyr J, Hill CJ, Jahangir M, Newton A, Petropoulos CJ, Huang W, Kurt-Yilmaz N, Schiffer CA, Ali A.
Matthew AN, et al. Among authors: zephyr j.
J Med Chem. 2017 Jul 13;60(13):5699-5716. doi: 10.1021/acs.jmedchem.7b00426. Epub 2017 Jun 19.
J Med Chem. 2017.
PMID: 28594175
Free PMC article.
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Avoiding Drug Resistance by Substrate Envelope-Guided Design: Toward Potent and Robust HCV NS3/4A Protease Inhibitors.
Matthew AN, Zephyr J, Nageswara Rao D, Henes M, Kamran W, Kosovrasti K, Hedger AK, Lockbaum GJ, Timm J, Ali A, Kurt Yilmaz N, Schiffer CA.
Matthew AN, et al. Among authors: zephyr j.
mBio. 2020 Mar 31;11(2):e00172-20. doi: 10.1128/mBio.00172-20.
mBio. 2020.
PMID: 32234812
Free PMC article.
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Discovery of Quinoxaline-Based P1-P3 Macrocyclic NS3/4A Protease Inhibitors with Potent Activity against Drug-Resistant Hepatitis C Virus Variants.
Nageswara Rao D, Zephyr J, Henes M, Chan ET, Matthew AN, Hedger AK, Conway HL, Saeed M, Newton A, Petropoulos CJ, Huang W, Kurt Yilmaz N, Schiffer CA, Ali A.
Nageswara Rao D, et al. Among authors: zephyr j.
J Med Chem. 2021 Aug 26;64(16):11972-11989. doi: 10.1021/acs.jmedchem.1c00554. Epub 2021 Aug 18.
J Med Chem. 2021.
PMID: 34405680
Free PMC article.
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Viral proteases: Structure, mechanism and inhibition.
Zephyr J, Kurt Yilmaz N, Schiffer CA.
Zephyr J, et al.
Enzymes. 2021;50:301-333. doi: 10.1016/bs.enz.2021.09.004. Epub 2021 Nov 17.
Enzymes. 2021.
PMID: 34861941
Free PMC article.
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Deciphering the Molecular Mechanism of HCV Protease Inhibitor Fluorination as a General Approach to Avoid Drug Resistance.
Zephyr J, Nageswara Rao D, Vo SV, Henes M, Kosovrasti K, Matthew AN, Hedger AK, Timm J, Chan ET, Ali A, Kurt Yilmaz N, Schiffer CA.
Zephyr J, et al.
J Mol Biol. 2022 May 15;434(9):167503. doi: 10.1016/j.jmb.2022.167503. Epub 2022 Feb 17.
J Mol Biol. 2022.
PMID: 35183560
Free PMC article.
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Allosteric quinoxaline-based inhibitors of the flavivirus NS2B/NS3 protease.
Zephyr J, Rao DN, Johnson C, Shaqra AM, Nalivaika EA, Jordan A, Kurt Yilmaz N, Ali A, Schiffer CA.
Zephyr J, et al.
Bioorg Chem. 2023 Feb;131:106269. doi: 10.1016/j.bioorg.2022.106269. Epub 2022 Nov 19.
Bioorg Chem. 2023.
PMID: 36446201
Free PMC article.
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FruitFire: a luciferase based on a fruit fly metabolic enzyme.
Adams ST Jr, Zephyr J, Bohn MF, Schiffer CA, Miller SC.
Adams ST Jr, et al. Among authors: zephyr j.
bioRxiv [Preprint]. 2023 Jun 30:2023.06.30.547126. doi: 10.1101/2023.06.30.547126.
bioRxiv. 2023.
PMID: 37425765
Free PMC article.
Preprint.
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