Yous S - Search Results

1

Bitopic fluorescent antagonists of the A_2A adenosine receptor based on pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine functionalized congeners.

Duroux R, Ciancetta A, Mannes P, Yu J, Boyapati S, Gizewski E, Yous S, Ciruela F, Auchampach JA, Gao ZG, Jacobson KA. Duroux R, et al. Among authors: yous s. Medchemcomm. 2017 Aug 1;8(8):1659-1667. doi: 10.1039/C7MD00247E. Epub 2017 Jun 22. Medchemcomm. 2017. PMID: 29250307 Free PMC article.

2

Antagonists of the adenosine A_2A receptor based on a 2-arylbenzoxazole scaffold: Investigation of the C5- and C7-positions to enhance affinity.

Duroux R, Agouridas L, Renault N, El Bakali J, Furman C, Melnyk P, Yous S. Duroux R, et al. Among authors: yous s. Eur J Med Chem. 2018 Jan 20;144:151-163. doi: 10.1016/j.ejmech.2017.12.007. Epub 2017 Dec 5. Eur J Med Chem. 2018. PMID: 29268131 Free article.

3

Design, synthesis and evaluation of 2-aryl benzoxazoles as promising hit for the A_2A receptor.

Duroux R, Renault N, Cuelho JE, Agouridas L, Blum D, Lopes LV, Melnyk P, Yous S. Duroux R, et al. Among authors: yous s. J Enzyme Inhib Med Chem. 2017 Dec;32(1):850-864. doi: 10.1080/14756366.2017.1334648. J Enzyme Inhib Med Chem. 2017. PMID: 28661196 Free PMC article.

4

High ligand efficiency quinazoline compounds as novel A_2A adenosine receptor antagonists.

Bolteau R, Duroux R, Laversin A, Vreulz B, Shiriaeva A, Stauch B, Han GW, Cherezov V, Renault N, Barczyk A, Ravez S, Coevoet M, Melnyk P, Liberelle M, Yous S. Bolteau R, et al. Among authors: yous s. Eur J Med Chem. 2022 Nov 5;241:114620. doi: 10.1016/j.ejmech.2022.114620. Epub 2022 Jul 22. Eur J Med Chem. 2022. PMID: 35933788

5

Design and synthesis of 2,6-disubstituted-8-amino imidazo[1,2a]pyridines, a promising privileged structure.

Boulahjar R, Rincon Arias A, Bolteau R, Renault N, Coevoet M, Barczyk A, Duroux R, Yous S, Melnyk P, Agouridas L. Boulahjar R, et al. Among authors: yous s. Bioorg Med Chem. 2018 Jul 23;26(12):3296-3307. doi: 10.1016/j.bmc.2018.04.057. Epub 2018 Apr 30. Bioorg Med Chem. 2018. PMID: 29753566 Free article.

6

Synthesis and biological evaluation of new naphtho- and quinolinocyclopentane derivatives as potent melatoninergic (MT₁/MT₂) and serotoninergic (5-HT_2C) dual ligands.

Duroux R, Rami M, Landagaray E, Ettaoussi M, Caignard DH, Delagrange P, Melnyk P, Yous S. Duroux R, et al. Among authors: yous s. Eur J Med Chem. 2017 Dec 1;141:552-566. doi: 10.1016/j.ejmech.2017.10.025. Epub 2017 Oct 12. Eur J Med Chem. 2017. PMID: 29102176

7

Melatonergic ligands: Design, synthesis and pharmacological evaluation of novel series of naphthofuranic derivatives.

Landagaray E, Ettaoussi M, Duroux R, Boutin JA, Caignard DH, Delagrange P, Melnyk P, Berthelot P, Yous S. Landagaray E, et al. Among authors: yous s. Eur J Med Chem. 2016 Feb 15;109:360-70. doi: 10.1016/j.ejmech.2015.12.047. Epub 2015 Dec 29. Eur J Med Chem. 2016. PMID: 26820449

8

Design and synthesis of naphthalenic derivatives as new ligands at the melatonin binding site MT3.

Leclerc V, Ettaoussi M, Rami M, Farce A, Boutin JA, Delagrange P, Caignard DH, Renard P, Berthelot P, Yous S. Leclerc V, et al. Among authors: yous s. Eur J Med Chem. 2011 May;46(5):1622-9. doi: 10.1016/j.ejmech.2011.02.010. Epub 2011 Feb 15. Eur J Med Chem. 2011. PMID: 21377769

9

Publisher Correction: Structural basis of ligand recognition at the human MT₁ melatonin receptor.

Stauch B, Johansson LC, McCorvy JD, Patel N, Han GW, Huang XP, Gati C, Batyuk A, Slocum ST, Ishchenko A, Brehm W, White TA, Michaelian N, Madsen C, Zhu L, Grant TD, Grandner JM, Shiriaeva A, Olsen RHJ, Tribo AR, Yous S, Stevens RC, Weierstall U, Katritch V, Roth BL, Liu W, Cherezov V. Stauch B, et al. Among authors: yous s. Nature. 2019 May;569(7756):E6. doi: 10.1038/s41586-019-1209-0. Nature. 2019. PMID: 31048811

10

Carbazole scaffolds in cancer therapy: a review from 2012 to 2018.

Issa S, Prandina A, Bedel N, Rongved P, Yous S, Le Borgne M, Bouaziz Z. Issa S, et al. Among authors: yous s. J Enzyme Inhib Med Chem. 2019 Dec;34(1):1321-1346. doi: 10.1080/14756366.2019.1640692. J Enzyme Inhib Med Chem. 2019. PMID: 31328585 Free PMC article. Review.

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