Rational design, synthesis, and structure-activity relationships of novel factor Xa inhibitors: (2-substituted-4-amidinophenyl)pyruvic and -propionic acids.
Sagi K, Nakagawa T, Yamanashi M, Makino S, Takahashi M, Takayanagi M, Takenaka K, Suzuki N, Oono S, Kataoka N, Ishikawa K, Shima S, Fukuda Y, Kayahara T, Takehana S, Shima Y, Tashiro K, Yamamoto H, Yoshimoto R, Iwata S, Tsuji T, Sakurai K, Shoji M.
Sagi K, et al. Among authors: yamanashi m.
J Med Chem. 2003 May 8;46(10):1845-57. doi: 10.1021/jm020485x.
J Med Chem. 2003.
PMID: 12723948