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Potent leads based on CA-19L, an anti-HIV active HIV-1 capsid fragment.
Tsuji K, Wang R, Kobayakawa T, Owusu KB, Fujino M, Kaneko M, Yamamoto N, Murakami T, Tamamura H. Tsuji K, et al. Among authors: yamamoto n. Bioorg Med Chem. 2021 Jan 15;30:115923. doi: 10.1016/j.bmc.2020.115923. Epub 2020 Dec 7. Bioorg Med Chem. 2021. PMID: 33316719
Pharmacophore-based small molecule CXCR4 ligands.
Narumi T, Tanaka T, Hashimoto C, Nomura W, Aikawa H, Sohma A, Itotani K, Kawamata M, Murakami T, Yamamoto N, Tamamura H. Narumi T, et al. Among authors: yamamoto n. Bioorg Med Chem Lett. 2012 Jun 15;22(12):4169-72. doi: 10.1016/j.bmcl.2012.04.032. Epub 2012 Apr 20. Bioorg Med Chem Lett. 2012. PMID: 22579418
Multimerized CHR-derived peptides as HIV-1 fusion inhibitors.
Nomura W, Hashimoto C, Suzuki T, Ohashi N, Fujino M, Murakami T, Yamamoto N, Tamamura H. Nomura W, et al. Among authors: yamamoto n. Bioorg Med Chem. 2013 Aug 1;21(15):4452-8. doi: 10.1016/j.bmc.2013.05.060. Epub 2013 Jun 5. Bioorg Med Chem. 2013. PMID: 23800723 Free article.
Anti-HIV-1 peptide derivatives based on the HIV-1 Co-receptor CXCR4.
Hashimoto C, Nomura W, Narumi T, Fujino M, Tsutsumi H, Haseyama M, Yamamoto N, Murakami T, Tamamura H. Hashimoto C, et al. Among authors: yamamoto n. ChemMedChem. 2013 Oct;8(10):1668-72. doi: 10.1002/cmdc.201300289. Epub 2013 Aug 23. ChemMedChem. 2013. PMID: 24039179
CXCR4-derived synthetic peptides inducing anti-HIV-1 antibodies.
Hashimoto C, Nomura W, Narumi T, Fujino M, Nakahara T, Yamamoto N, Murakami T, Tamamura H. Hashimoto C, et al. Among authors: yamamoto n. Bioorg Med Chem. 2013 Nov 15;21(22):6878-85. doi: 10.1016/j.bmc.2013.09.037. Epub 2013 Sep 21. Bioorg Med Chem. 2013. PMID: 24119449
Development of anti-HIV peptides based on a viral capsid protein.
Mizuguchi T, Ohashi N, Matsumoto D, Hashimoto C, Nomura W, Yamamoto N, Murakami T, Tamamura H. Mizuguchi T, et al. Among authors: yamamoto n. Biopolymers. 2017 Jan;108(1). doi: 10.1002/bip.22920. Biopolymers. 2017. PMID: 27428649
Design, synthesis and biological evaluation of low molecular weight CXCR4 ligands.
Sakyiamah MM, Kobayakawa T, Fujino M, Konno M, Narumi T, Tanaka T, Nomura W, Yamamoto N, Murakami T, Tamamura H. Sakyiamah MM, et al. Among authors: yamamoto n. Bioorg Med Chem. 2019 Mar 15;27(6):1130-1138. doi: 10.1016/j.bmc.2019.02.013. Epub 2019 Feb 6. Bioorg Med Chem. 2019. PMID: 30772128
6,235 results