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Synthesis, computational and experimental pharmacological studies for (thio)ether-triazine 5-HT6R ligands with noticeable action on AChE/BChE and chalcogen-dependent intrinsic activity in search for new class of drugs against Alzheimer's disease.
Eur J Med Chem. 2023 Nov 5;259:115695. doi: 10.1016/j.ejmech.2023.115695. Epub 2023 Jul 30.
Eur J Med Chem. 2023.
PMID: 37567058
Free article.
An exit beyond the pharmacophore model for 5-HT6R agents - a new strategy to gain dual 5-HT6/5-HT2A action for triazine derivatives with procognitive potential.
Kucwaj-Brysz K, Ali W, Kurczab R, Sudoł-Tałaj S, Wilczyńska-Zawal N, Jastrzębska-Więsek M, Satała G, Mordyl B, Żesławska E, Agnieszka-Olejarz-Maciej, Czarnota K, Latacz G, Partyka A, Wesołowska A, Nitek W, Handzlik J.
Kucwaj-Brysz K, et al. Among authors: wilczynska zawal n.
Bioorg Chem. 2022 Apr;121:105695. doi: 10.1016/j.bioorg.2022.105695. Epub 2022 Feb 19.
Bioorg Chem. 2022.
PMID: 35228010
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The Phenoxyalkyltriazine Antagonists for 5-HT6 Receptor with Promising Procognitive and Pharmacokinetic Properties In Vivo in Search for a Novel Therapeutic Approach to Dementia Diseases.
Sudoł S, Cios A, Jastrzębska-Więsek M, Honkisz-Orzechowska E, Mordyl B, Wilczyńska-Zawal N, Satała G, Kucwaj-Brysz K, Partyka A, Latacz G, Olejarz-Maciej A, Wesołowska A, Handzlik J.
Sudoł S, et al. Among authors: wilczynska zawal n.
Int J Mol Sci. 2021 Oct 5;22(19):10773. doi: 10.3390/ijms221910773.
Int J Mol Sci. 2021.
PMID: 34639113
Free PMC article.
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Effect of 5-HT6 Receptor Ligands Combined with Haloperidol or Risperidone on Antidepressant-/Anxiolytic-Like Behavior and BDNF Regulation in Hippocampus and Prefrontal Cortex of Rats.
Wesołowska A, Rychtyk J, Gdula-Argasińska J, Górecka K, Wilczyńska-Zawal N, Jastrzębska-Więsek M, Partyka A.
Wesołowska A, et al. Among authors: wilczynska zawal n.
Neuropsychiatr Dis Treat. 2021 Jun 25;17:2105-2127. doi: 10.2147/NDT.S309818. eCollection 2021.
Neuropsychiatr Dis Treat. 2021.
PMID: 34211274
Free PMC article.
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Selective 5-HT6 Receptor Ligands (Agonist and Antagonist) Show Different Effects on Antipsychotic Drug-Induced Metabolic Dysfunctions in Rats.
Partyka A, Górecka K, Gdula-Argasińska J, Wilczyńska-Zawal N, Jastrzębska-Więsek M, Wesołowska A.
Partyka A, et al. Among authors: wilczynska zawal n.
Pharmaceuticals (Basel). 2023 Jan 20;16(2):154. doi: 10.3390/ph16020154.
Pharmaceuticals (Basel). 2023.
PMID: 37259305
Free PMC article.
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First-in-Class Selenium-Containing Potent Serotonin Receptor 5-HT6 Agents with a Beneficial Neuroprotective Profile against Alzheimer's Disease.
Pyka P, Haberek W, Więcek M, Szymanska E, Ali W, Cios A, Jastrzębska-Więsek M, Satała G, Podlewska S, Di Giacomo S, Di Sotto A, Garbo S, Karcz T, Lambona C, Marocco F, Latacz G, Sudoł-Tałaj S, Mordyl B, Głuch-Lutwin M, Siwek A, Czarnota-Łydka K, Gogola D, Olejarz-Maciej A, Wilczyńska-Zawal N, Honkisz-Orzechowska E, Starek M, Dąbrowska M, Kucwaj-Brysz K, Fioravanti R, Nasim MJ, Hittinger M, Partyka A, Wesołowska A, Battistelli C, Zwergel C, Handzlik J.
Pyka P, et al. Among authors: wilczynska zawal n.
J Med Chem. 2024 Jan 25;67(2):1580-1610. doi: 10.1021/acs.jmedchem.3c02148. Epub 2024 Jan 8.
J Med Chem. 2024.
PMID: 38190615
Free PMC article.
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Hydrophobicity modulation via the substituents at positions 2 and 4 of 1,3,5-triazine to enhance therapeutic ability against Alzheimer's disease for potent serotonin 5-HT6R agents.
Sudoł-Tałaj S, Kucwaj-Brysz K, Podlewska S, Kurczab R, Satała G, Mordyl B, Głuch-Lutwin M, Wilczyńska-Zawal N, Jastrzębska-Więsek M, Czarnota-Łydka K, Kurowska K, Kubacka M, Żesławska E, Nitek W, Olejarz-Maciej A, Doroz-Płonka A, Partyka A, Latacz G, Wesołowska A, Handzlik J.
Sudoł-Tałaj S, et al. Among authors: wilczynska zawal n.
Eur J Med Chem. 2023 Nov 15;260:115756. doi: 10.1016/j.ejmech.2023.115756. Epub 2023 Aug 24.
Eur J Med Chem. 2023.
PMID: 37657272
Free article.
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