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Discovery and Crystallographic Studies of Nonpeptidic Piperazine Derivatives as Covalent SARS-CoV-2 Main Protease Inhibitors.
J Med Chem. 2022 Dec 22;65(24):16902-16917. doi: 10.1021/acs.jmedchem.2c01716. Epub 2022 Dec 7.
J Med Chem. 2022.
PMID: 36475694
Discovery and Crystallographic Studies of Trisubstituted Piperazine Derivatives as Non-Covalent SARS-CoV-2 Main Protease Inhibitors with High Target Specificity and Low Toxicity.
Gao S, Sylvester K, Song L, Claff T, Jing L, Woodson M, Weiße RH, Cheng Y, Schäkel L, Petry M, Gütschow M, Schiedel AC, Sträter N, Kang D, Xu S, Toth K, Tavis J, Tollefson AE, Müller CE, Liu X, Zhan P.
Gao S, et al. Among authors: weisse rh.
J Med Chem. 2022 Oct 13;65(19):13343-13364. doi: 10.1021/acs.jmedchem.2c01146. Epub 2022 Sep 15.
J Med Chem. 2022.
PMID: 36107752
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Structural and Mechanistic Studies on Substrate and Stereoselectivity of the Indole Monooxygenase VpIndA1: New Avenues for Biocatalytic Epoxidations and Sulfoxidations.
Kratky J, Eggerichs D, Heine T, Hofmann S, Sowa P, Weiße RH, Tischler D, Sträter N.
Kratky J, et al. Among authors: weisse rh.
Angew Chem Int Ed Engl. 2023 Apr 17;62(17):e202300657. doi: 10.1002/anie.202300657. Epub 2023 Mar 16.
Angew Chem Int Ed Engl. 2023.
PMID: 36762980
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Crystal structure of adenosine A2A receptor in complex with clinical candidate Etrumadenant reveals unprecedented antagonist interaction.
Claff T, Schlegel JG, Voss JH, Vaaßen VJ, Weiße RH, Cheng RKY, Markovic-Mueller S, Bucher D, Sträter N, Müller CE.
Claff T, et al. Among authors: weisse rh.
Commun Chem. 2023 Jun 1;6(1):106. doi: 10.1038/s42004-023-00894-6.
Commun Chem. 2023.
PMID: 37264098
Free PMC article.
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The dimerized pentraxin-like domain of the adhesion G protein-coupled receptor 112 (ADGRG4) suggests function in sensing mechanical forces.
Kieslich B, Weiße RH, Brendler J, Ricken A, Schöneberg T, Sträter N.
Kieslich B, et al. Among authors: weisse rh.
J Biol Chem. 2023 Dec;299(12):105356. doi: 10.1016/j.jbc.2023.105356. Epub 2023 Oct 18.
J Biol Chem. 2023.
PMID: 37863265
Free PMC article.
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Design, Synthesis, and Biological Evaluation of Trisubstituted Piperazine Derivatives as Noncovalent Severe Acute Respiratory Syndrome Coronavirus 2 Main Protease Inhibitors with Improved Antiviral Activity and Favorable Druggability.
Gao S, Song L, Sylvester K, Mercorelli B, Loregian A, Toth K, Weiße RH, Useini A, Sträter N, Yang M, Ye B, Tollefson AE, Müller CE, Liu X, Zhan P.
Gao S, et al. Among authors: weisse rh.
J Med Chem. 2023 Dec 14;66(23):16426-16440. doi: 10.1021/acs.jmedchem.3c01876. Epub 2023 Nov 22.
J Med Chem. 2023.
PMID: 37992202
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Structure of NDP-forming Acetyl-CoA synthetase ACD1 reveals a large rearrangement for phosphoryl transfer.
Weiße RH, Faust A, Schmidt M, Schönheit P, Scheidig AJ.
Weiße RH, et al.
Proc Natl Acad Sci U S A. 2016 Feb 2;113(5):E519-28. doi: 10.1073/pnas.1518614113. Epub 2016 Jan 19.
Proc Natl Acad Sci U S A. 2016.
PMID: 26787904
Free PMC article.
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