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71 results

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Page 1
Isoxazolo(aza)naphthoquinones: a new class of cytotoxic Hsp90 inhibitors.
Bargiotti A, Musso L, Dallavalle S, Merlini L, Gallo G, Ciacci A, Giannini G, Cabri W, Penco S, Vesci L, Castorina M, Milazzo FM, Cervoni ML, Barbarino M, Pisano C, Giommarelli C, Zuco V, De Cesare M, Zunino F. Bargiotti A, et al. Among authors: vesci l. Eur J Med Chem. 2012 Jul;53:64-75. doi: 10.1016/j.ejmech.2012.03.036. Epub 2012 Mar 28. Eur J Med Chem. 2012. PMID: 22538015
Synthesis and evaluation of new Hsp90 inhibitors based on a 1,4,5-trisubstituted 1,2,3-triazole scaffold.
Taddei M, Ferrini S, Giannotti L, Corsi M, Manetti F, Giannini G, Vesci L, Milazzo FM, Alloatti D, Guglielmi MB, Castorina M, Cervoni ML, Barbarino M, Foderà R, Carollo V, Pisano C, Armaroli S, Cabri W. Taddei M, et al. Among authors: vesci l. J Med Chem. 2014 Mar 27;57(6):2258-74. doi: 10.1021/jm401536b. Epub 2014 Mar 17. J Med Chem. 2014. PMID: 24588105
A novel atypical retinoid endowed with proapoptotic and antitumor activity.
Cincinelli R, Dallavalle S, Merlini L, Penco S, Pisano C, Carminati P, Giannini G, Vesci L, Gaetano C, Illy B, Zuco V, Supino R, Zunino F. Cincinelli R, et al. Among authors: vesci l. J Med Chem. 2003 Mar 13;46(6):909-12. doi: 10.1021/jm025593y. J Med Chem. 2003. PMID: 12620066
Natural and semisynthetic azaphilones as a new scaffold for Hsp90 inhibitors.
Musso L, Dallavalle S, Merlini L, Bava A, Nasini G, Penco S, Giannini G, Giommarelli C, De Cesare A, Zuco V, Vesci L, Pisano C, Castorina M, Milazzo F, Cervoni ML, Dal Piaz F, De Tommasi N, Zunino F. Musso L, et al. Among authors: vesci l. Bioorg Med Chem. 2010 Aug 15;18(16):6031-43. doi: 10.1016/j.bmc.2010.06.068. Epub 2010 Jul 1. Bioorg Med Chem. 2010. PMID: 20655237
Novel 3,4-isoxazolediamides as potent inhibitors of chaperone heat shock protein 90.
Baruchello R, Simoni D, Grisolia G, Barbato G, Marchetti P, Rondanin R, Mangiola S, Giannini G, Brunetti T, Alloatti D, Gallo G, Ciacci A, Vesci L, Castorina M, Milazzo FM, Cervoni ML, Guglielmi MB, Barbarino M, Foderà R, Pisano C, Cabri W. Baruchello R, et al. Among authors: vesci l. J Med Chem. 2011 Dec 22;54(24):8592-604. doi: 10.1021/jm201155e. Epub 2011 Nov 23. J Med Chem. 2011. PMID: 22066525
New retinoid derivatives as back-ups of Adarotene.
Giannini G, Brunetti T, Battistuzzi G, Alloatti D, Quattrociocchi G, Cima MG, Merlini L, Dallavalle S, Cincinelli R, Nannei R, Vesci L, Bucci F, Foderà R, Guglielmi MB, Pisano C, Cabri W. Giannini G, et al. Among authors: vesci l. Bioorg Med Chem. 2012 Apr 1;20(7):2405-15. doi: 10.1016/j.bmc.2012.01.042. Epub 2012 Feb 6. Bioorg Med Chem. 2012. PMID: 22365912
71 results