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Enzymatic Preparation of 2'-5',3'-5'-Cyclic Dinucleotides, Their Binding Properties to Stimulator of Interferon Genes Adaptor Protein, and Structure/Activity Correlations.
Novotná B, Vaneková L, Zavřel M, Buděšínský M, Dejmek M, Smola M, Gutten O, Tehrani ZA, Pimková Polidarová M, Brázdová A, Liboska R, Štěpánek I, Vavřina Z, Jandušík T, Nencka R, Rulíšek L, Bouřa E, Brynda J, Páv O, Birkuš G. Novotná B, et al. Among authors: vavrina z. J Med Chem. 2019 Dec 12;62(23):10676-10690. doi: 10.1021/acs.jmedchem.9b01062. Epub 2019 Nov 27. J Med Chem. 2019. PMID: 31715099
Enzymatic Synthesis of 3'-5', 3'-5' Cyclic Dinucleotides, Their Binding Properties to the Stimulator of Interferon Genes Adaptor Protein, and Structure/Activity Correlations.
Novotná B, Holá L, Staś M, Gutten O, Smola M, Zavřel M, Vavřina Z, Buděšínský M, Liboska R, Chevrier F, Dobiaš J, Boura E, Rulíšek L, Birkuš G. Novotná B, et al. Among authors: vavrina z. Biochemistry. 2021 Dec 7;60(48):3714-3727. doi: 10.1021/acs.biochem.1c00692. Epub 2021 Nov 17. Biochemistry. 2021. PMID: 34788017
5'-Phosphonate modified oligoadenylates as potent activators of human RNase L.
Lášek T, Petrová M, Košiová I, Šimák O, Buděšínský M, Kozák J, Snášel J, Vavřina Z, Birkuš G, Rosenberg I, Páv O. Lášek T, et al. Among authors: vavrina z. Bioorg Med Chem. 2022 Feb 15;56:116632. doi: 10.1016/j.bmc.2022.116632. Epub 2022 Jan 19. Bioorg Med Chem. 2022. PMID: 35078032
Corrigendum to "5'-Phosphonate modified oligoadenylates as potent activators of human RNase L" [Bioorg. Med. Chem. 56 (2022) 116632].
Lášek T, Petrová M, Košiová I, Šimák O, Buděšínský M, Kozák J, Snášel J, Vavřina Z, Birkuš G, Rosenberg I, Páv O. Lášek T, et al. Among authors: vavrina z. Bioorg Med Chem. 2022 Mar 15;58:116654. doi: 10.1016/j.bmc.2022.116654. Epub 2022 Feb 10. Bioorg Med Chem. 2022. PMID: 35153131 No abstract available.
Design, Synthesis, and Biochemical and Biological Evaluation of Novel 7-Deazapurine Cyclic Dinucleotide Analogues as STING Receptor Agonists.
Vavřina Z, Perlíková P, Milisavljević N, Chevrier F, Smola M, Smith J, Dejmek M, Havlíček V, Buděšínský M, Liboska R, Vaneková L, Brynda J, Boura E, Řezáčová P, Hocek M, Birkuš G. Vavřina Z, et al. J Med Chem. 2022 Oct 27;65(20):14082-14103. doi: 10.1021/acs.jmedchem.2c01305. Epub 2022 Oct 6. J Med Chem. 2022. PMID: 36201304 Free PMC article.
Vinylphosphonate-based cyclic dinucleotides enhance STING-mediated cancer immunotherapy.
Dejmek M, Brazdova A, Otava T, Polidarova MP, Klíma M, Smola M, Vavrina Z, Buděšínský M, Dračínský M, Liboska R, Boura E, Birkuš G, Nencka R. Dejmek M, et al. Among authors: vavrina z. Eur J Med Chem. 2023 Nov 5;259:115685. doi: 10.1016/j.ejmech.2023.115685. Epub 2023 Jul 26. Eur J Med Chem. 2023. PMID: 37567057 Free article.