Potent Inhibition of SARS-CoV-2 nsp14 N7-Methyltransferase by Sulfonamide-Based Bisubstrate Analogues.
Ahmed-Belkacem R, Hausdorff M, Delpal A, Sutto-Ortiz P, Colmant AMG, Touret F, Ogando NS, Snijder EJ, Canard B, Coutard B, Vasseur JJ, Decroly E, Debart F.
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J Med Chem. 2022 Apr 28;65(8):6231-6249. doi: 10.1021/acs.jmedchem.2c00120. Epub 2022 Apr 19.
J Med Chem. 2022.
PMID: 35439007