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The First Enantioselective Total Synthesis of (-)-trans-Dihydronarciclasine.
J Nat Prod. 2017 Jun 23;80(6):1909-1917. doi: 10.1021/acs.jnatprod.7b00208. Epub 2017 Jun 5.
J Nat Prod. 2017.
PMID: 28581297
Free article.
(±)-trans-Dihydronarciclasine and (±)-trans-dihydrolycoricidine analogues modified in their ring A: Evaluation of their anticancer activity and a SAR study.
Varró G, Pálchuber P, Pogrányi B, Simon A, Hegedűs L, Kádas I.
Varró G, et al.
Eur J Med Chem. 2019 Jul 1;173:76-89. doi: 10.1016/j.ejmech.2019.04.010. Epub 2019 Apr 8.
Eur J Med Chem. 2019.
PMID: 30986573
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Stereoselective synthesis of trans-dihydronarciclasine derivatives containing a 1,4-benzodioxane moiety.
Varró G, Pogrányi B, Grün A, Simon A, Hegedűs L, Kádas I.
Varró G, et al.
Monatsh Chem. 2018;149(12):2265-2285. doi: 10.1007/s00706-018-2287-7. Epub 2018 Oct 26.
Monatsh Chem. 2018.
PMID: 32214482
Free PMC article.
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Multiparameter Optimization of Naphthyridine Derivatives as Selective α5-GABAA Receptor Negative Allosteric Modulators.
Szabó G, Éliás O, Erdélyi P, Potor A, Túrós GI, Károlyi BI, Varró G, Vaskó ÁG, Bata I, Kapus GL, Dohányos Z, Bobok AÁ, Fodor L, Thán M, Vastag M, Komlódi Z, Soukupné Kedves RÉ, Makó É, Süveges B, Greiner I.
Szabó G, et al. Among authors: varro g.
J Med Chem. 2022 Jun 9;65(11):7876-7895. doi: 10.1021/acs.jmedchem.2c00414. Epub 2022 May 18.
J Med Chem. 2022.
PMID: 35584373
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