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Synthesis of Prostate-Specific Membrane Antigen-Targeted Bimodal Conjugates of Cytotoxic Agents and Antiandrogens and Their Comparative Assessment with Monoconjugates.
Int J Mol Sci. 2023 Jul 11;24(14):11327. doi: 10.3390/ijms241411327.
Int J Mol Sci. 2023.
PMID: 37511087
Free PMC article.
Synthesis and Preclinical Evaluation of Small-Molecule Prostate-Specific Membrane Antigen-Targeted Abiraterone Conjugate.
Machulkin AE, Nimenko EA, Zyk NU, Uspenskaia AA, Smirnova GB, Khan II, Pokrovsky VS, Vaneev AN, Timoshenko RV, Mamed-Nabizade VV, Zavertkina MV, Erofeev A, Gorelkin P, Majouga AG, Zyk NV, Khazanova ES, Beloglazkina EK.
Machulkin AE, et al. Among authors: uspenskaia aa.
Molecules. 2022 Dec 12;27(24):8795. doi: 10.3390/molecules27248795.
Molecules. 2022.
PMID: 36557929
Free PMC article.
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Fluorescent Conjugates Based on Prostate-Specific Membrane Antigen Ligands as an Effective Visualization Tool for Prostate Cancer.
Uspenskaia AA, Krasnikov PA, Majouga AG, Beloglazkina EK, Machulkin AE.
Uspenskaia AA, et al.
Biochemistry (Mosc). 2023 Jul;88(7):953-967. doi: 10.1134/S0006297923070088.
Biochemistry (Mosc). 2023.
PMID: 37751866
Review.
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