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CDK inhibitors: from the bench to clinical trials.
Rizzolio F, Tuccinardi T, Caligiuri I, Lucchetti C, Giordano A. Rizzolio F, et al. Among authors: tuccinardi t. Curr Drug Targets. 2010 Mar;11(3):279-90. doi: 10.2174/138945010790711978. Curr Drug Targets. 2010. PMID: 20210753 Review.
Identification of new Fyn kinase inhibitors using a FLAP-based approach.
Poli G, Tuccinardi T, Rizzolio F, Caligiuri I, Botta L, Granchi C, Ortore G, Minutolo F, Schenone S, Martinelli A. Poli G, et al. Among authors: tuccinardi t. J Chem Inf Model. 2013 Oct 28;53(10):2538-47. doi: 10.1021/ci4002553. Epub 2013 Sep 16. J Chem Inf Model. 2013. PMID: 24001328
Identification and characterization of a new reversible MAGL inhibitor.
Tuccinardi T, Granchi C, Rizzolio F, Caligiuri I, Battistello V, Toffoli G, Minutolo F, Macchia M, Martinelli A. Tuccinardi T, et al. Bioorg Med Chem. 2014 Jul 1;22(13):3285-91. doi: 10.1016/j.bmc.2014.04.057. Epub 2014 May 6. Bioorg Med Chem. 2014. PMID: 24853323
Highly selective salicylketoxime-based estrogen receptor β agonists display antiproliferative activities in a glioma model.
Paterni I, Bertini S, Granchi C, Tuccinardi T, Macchia M, Martinelli A, Caligiuri I, Toffoli G, Rizzolio F, Carlson KE, Katzenellenbogen BS, Katzenellenbogen JA, Minutolo F. Paterni I, et al. Among authors: tuccinardi t. J Med Chem. 2015 Feb 12;58(3):1184-94. doi: 10.1021/jm501829f. Epub 2015 Jan 14. J Med Chem. 2015. PMID: 25559213 Free PMC article.
Cyclic Ketoximes as Estrogen Receptor β Selective Agonists.
Granchi C, Lapillo M, Spena CR, Rizzolio F, Tuccinardi T, Martin TA, Carlson KE, Katzenellenbogen JA, Minutolo F. Granchi C, et al. Among authors: tuccinardi t. ChemMedChem. 2016 Aug 19;11(16):1752-61. doi: 10.1002/cmdc.201600140. Epub 2016 May 2. ChemMedChem. 2016. PMID: 27135651 Free PMC article.
Structural Optimization of 4-Chlorobenzoylpiperidine Derivatives for the Development of Potent, Reversible, and Selective Monoacylglycerol Lipase (MAGL) Inhibitors.
Granchi C, Rizzolio F, Palazzolo S, Carmignani S, Macchia M, Saccomanni G, Manera C, Martinelli A, Minutolo F, Tuccinardi T. Granchi C, et al. Among authors: tuccinardi t. J Med Chem. 2016 Nov 23;59(22):10299-10314. doi: 10.1021/acs.jmedchem.6b01459. Epub 2016 Nov 14. J Med Chem. 2016. PMID: 27809504
Bottom-up synthesis of carbon nanoparticles with higher doxorubicin efficacy.
Bayda S, Hadla M, Palazzolo S, Kumar V, Caligiuri I, Ambrosi E, Pontoglio E, Agostini M, Tuccinardi T, Benedetti A, Riello P, Canzonieri V, Corona G, Toffoli G, Rizzolio F. Bayda S, et al. Among authors: tuccinardi t. J Control Release. 2017 Feb 28;248:144-152. doi: 10.1016/j.jconrel.2017.01.022. Epub 2017 Jan 14. J Control Release. 2017. PMID: 28093297 Free article.
216 results